ELB-139 NEW
| Price | $293 | $436 | $722 |
| Package | 1mg | 2mg | 5mg |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2025-09-18 |
Product Details
| Product Name: ELB-139 | CAS No.: 188116-08-7 |
| Purity: 100.00% | Supply Ability: 10g |
| Release date: 2025/09/18 |
Product Introduction
Bioactivity
| Name | ELB-139 |
| Description | ELB-139 is a GABAA receptor agonist that can be used to study depression and epilepsy. |
| In vitro | The IC(50) for the binding site of ELB139 to flunitrazepam in rat forebrain cortical membranes was 1390 nM.In rat hippocampal neurons, ELB139 potentiated GABA-induced currents without maximal effects of diazepam, suggesting partial benzodiazepine agonism. [5] |
| In vivo | ELB139 (10 and 30 mg/kg orally) was active in three different animal models of anxiety in elevated plus maze, light and dark boxes, and Vogel conflict tests. [5] |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Keywords | GABAReceptor | GABAA | GABA Receptor | ELB-139 |
| Inhibitors Related | Valproic acid sodium salt | DL-Menthol | Urethane | p-Hydroxybenzaldehyde | Penicillin G sodium salt | Valproic Acid | Halothane | Chlorothymol | Piperazine citrate | Riluzole | (-)-α-Pinene | Methionine |
| Related Compound Libraries | Pain-Related Compound Library | Bioactive Compound Library | Neuronal Signaling Compound Library | Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | Ion Channel Targeted Library |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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United States- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, MA
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