Pilsicainide NEW
| Price | $1520 | $1980 | $2500 |
| Package | 25mg | 50mg | 100mg |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2025-10-27 |
Product Details
| Product Name: Pilsicainide | CAS No.: 88069-67-4 |
| Supply Ability: 10g | Release date: 2025/10/27 |
Product Introduction
Bioactivity
| Name | Pilsicainide |
| Description | Pilsicainide (SUN 1165 free acid) is a potent class Ic antiarrhythmic agent and a sodium channel blocker[1][2]. |
| In vitro | Pilsicainide (SUN 1165 free acid; 10-200 μg/mL) dose-dependently reduces the peak amplitude of the net inward current, with an IC50 of 29.2 μg/mL in levo-thyroxine (T4)-treated rat atrial cells [1]. |
| In vivo | Pilsicainide (SUN 1165 free acid; 2 mg/kg; i.v.; once) significantly reduces conduction velocity in the atrium of T4-treated male Sprague-Dawley rats (weighing 200-220 g) by decreasing Max dV/dt and net inward current, and altering electrocardiographic parameters. Administered as a bolus into the right external carotid vein over two minutes, pilsicainide extends the QT interval at 15 and 60 minutes post-administration, decreases the durations of P wave and QRS complex, reduces action potential amplitudes (APA) and Max dV/dt, and lengthens action potential duration. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Inhibitors Related | Pramocaine hydrochloride | Phenytoin sodium | Procaine | Tetracaine hydrochloride | Lidocaine | Safinamide | Valproic Acid | L-Aspartic aicd sodium | Lidocaine hydrochloride | Mebeverine hydrochloride | Dibucaine | Ropivacaine hydrochloride |
Company Profile Introduction
TargetMol Chemicals Inc. is headquartered in Boston, MA, and specializes in products and services that serve the research needs of chemical and biological scientists worldwide. With a client base in 40+ countries, TargetMol has evolved into one of the biggest global research suppliers for compound libraries and small molecule compounds.
170+ Compound Libraries， 10000+ Noval Small Molecucles，16000+ Nature Compounds
TargetMol diligently updates and offers over 170 types of compound libraries and a wide range of high-quality research chemicals, including inhibitors, activators, natural products, peptides, antibodies , and novel life-science kits for laboratory and scientific use. In addition, our lab allows us to conduct CADD (computer-aided drug design) and chemical synthesis to meet the customization needs of our clients.
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United States- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, Massachusetts, USA
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