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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
1-phenylcyclopropane-1-sulfonamide 1-苯基环丙烷-1-磺酰胺 646051-96-9 详细
3-cyclohexyl-1H-indole-6-carboxylic acid 494799-17-6 详细
3-(4-fluorophenyl)oxetan-3-yl]methanamine 1260664-08-1 详细
4-[(S)-(3-propylimidazol-4-yl)methylsulfinyl]aniline 4-[(S)-(1-丙基-1H-咪唑-5-基)甲亚磺酰基]苯胺 497223-38-8 详细
trans-2-(4-ethoxy-3-fluoro-phenyl)cyclopropanamine;hydrochloride (1S,2R)-rel-2-(4-乙氧基-3-氟苯基)环丙烷-1-胺盐酸 2055841-15-9 详细
1-[6-(trifluoromethyl)-3-pyridyl]cyclopropanecarboxylic acid 1060811-01-9 详细
(5R,6S)-5,6-diphenylmorpholin-2-one 282735-66-4 详细
3-amino-1-(2-pyridyl)pyridin-2-one 1797435-79-0 详细
cis-3-hydroxy-3-phenyl-cyclobutanecarboxylic acid 1812175-28-2 详细
tert-butyl N-[1-(azetidin-3-yl)-4-piperidyl]carbamate;hydrochloride 2940938-63-4 详细
4-phenyloxane-4-carboxylic acid 182491-21-0 详细
(2S)-2-phenylmorpholine 74572-15-9 详细
6-bromo-5-(2-fluoro-4-nitrophenoxy)-1-methyl-1H-indazole 6-溴-5-(2-氟-4-硝基苯氧基)-1-甲基-1H-吲唑 1206800-24-9 详细
(3S)-3-benzyl-1-[(tert-butoxy)carbonyl]piperidine-3-carboxylic acid 170838-87-6 详细
4-amino-1-[(2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl]-1,2-dihydropyrimidin-2-one 4-氨基-1-[(2R,5S)-2-(羟甲基)-1,3-噁噻戊环-5-基]-1,2-二氢嘧啶-2-酮 134678-17-4 详细
2-(3-bromophenyl)-4,4-dimethyl-N-(propan-2-yl)-1,2,3,4-tetrahydroquinoline-6-sulfonamide 2-(3-溴苯基)-4,4-二甲基-N-(丙烷-2-基)-1,2,3,4-四氢喹啉-6-磺酰胺 1391609-03-2 详细
2-methoxy-4-{9-methyl-3,9-diazaspiro[5.5]undecan-3-yl}aniline 2-甲氧基-4-{9-甲基-3,9-二氮杂螺[5.5]十一烷-3-基}苯胺 1818847-36-7 详细
(1R,5S)-1-(4-bromophenyl)-3-azabicyclo[3.1.0]hexane 956037-89-1 详细
1-[3-fluoro-2-(trifluoromethyl)pyridine-4-carbonyl]piperidin-4-ol 1-[3-氟-2-(三氟甲基)吡啶-4-羰基]哌啶-4-醇 2126176-86-9 详细
4-bromo-2-[(trans-4-hydroxycyclohexyl)amino]benzonitrile 1008520-76-0 详细
(1R,2R)-2-amino-1,2-diphenylethan-1-ol (1R,2R)-2-氨基-1,2-二苯基乙烷-1-醇 88082-66-0 详细
tert-butyl 4-[cis-2-aminocyclohexyl]piperazine-1-carboxylate 叔-丁基 4-[顺-2-氨基环己基]哌嗪-1-甲酸基酯 2177263-19-1 详细
1-pyrrolidin-2-ylcyclopropanol 1784640-67-0 详细
6-phenyl-2-azaspiro[3.3]heptane;hydrochloride 2445478-10-2 详细
4-[trans-2-aminocyclopropyl]phenol 4-[(1R,2S)-rel-2-氨基环丙基]苯酚 104777-77-7 详细
cis-4-(3-amino-2,2,4,4-tetramethyl-cyclobutoxy)-2-chloro-benzonitrile;hydrochloride 2891581-06-7 详细
4-(1H-1,3-benzodiazol-2-yl)-1,2,5-oxadiazol-3-amine 4-(1H-1,3-苯并二唑-2-基)-1,2,5-噁二唑-3-胺 332026-86-5 详细
4-[(3-fluorophenyl)methoxy]-3-[(3-fluorophenyl)methyl]benzaldehyde 4-[(3-氟苯基)甲氧基]-3-[(3-氟苯基)甲基]苯(甲)醛 1000370-24-0 详细
2-chloro-4-(3-nitrophenoxy)thieno[3,2-d]pyrimidine 2-氯-4-(3-硝基苯氧基)噻吩并[3,2-d]嘧啶 1353553-07-7 详细
N-cyclopropyl-1H-indole-5-sulfonamide N-环丙基-1H-吲哚-5-磺酰胺 1860028-27-8 详细
1-(5-bromopyrimidin-2-yl)cyclopropan-1-amine hydrochloride 1-(5-溴嘧啶-2-基)环丙烷-1-胺盐酸 2055841-13-7 详细
4-(azetidin-1-yl)aniline 344405-51-2 详细
(3-phenyloxetan-3-yl)methanamine (3-苯基噁丁环烷-3-基)甲胺 497239-45-9 详细
tert-butyl 3-hydroxy-3-phenyl-azetidine-1-carboxylate 398489-25-3 详细
1-cyclopropyl-1H-pyrazol-4-amine 1240567-18-3 详细
(3S)-3-phenylpyrrolidine (3S)-3-苯基吡咯烷 62624-46-8 详细
ethyl 3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazole-5-carboxylate 1258269-03-2 详细
trans-2-(2-bromothiazol-5-yl)cyclopropanamine dihydrobromide (1S,2S)-rel-2-(2-溴-1,3-噻唑-5-基)环丙烷-1-胺二氢溴酸盐 2173052-92-9 详细
1-phenyl-4-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole 1002334-12-4 详细
tert-butyl N-[(1R,2S)-1-(cyclopropylsulfonylcarbamoyl)-2-vinyl-cyclopropyl]carbamate 630421-48-6 详细
1-[[2-fluoro-6-(trifluoromethyl)phenyl]methyl]-6-methyl-pyrimidine-2,4-dione 830346-47-9 详细
2-[1-(ethanesulfonyl)-3-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]azetidin-3-yl]acetonitrile 2-[1-(乙磺酰)-3-[4-(4,4,5,5-四甲基-1,3,2-二噁硼戊环-2-基)-1H-吡唑-1-基]吖丁啶-3-基]乙腈 1919837-50-5 详细
1-(azetidin-3-yl)-4-methylpiperazine trihydrochloride 1803590-57-9 详细
1-(azetidin-3-yl)azetidine;bis(2,2,2-trifluoroacetic acid) 1909335-95-0 详细
cis-4-(5-bromo-2-chloro-pyrrolo[2,3-d]pyrimidin-7-yl)cyclohexanol 2227199-18-8 详细
(5S)-5-[4-(trifluoromethyl)phenyl]morpholin-3-one 1344400-76-5 详细
(4-methoxycarbonyl-2,6-dimethyl-phenyl) 9,10-dihydroacridine-9-carboxylate 1536146-87-8 详细
4-{6-[(tert-butoxy)carbonyl]-2,6-diazaspiro[3.3]heptan-2-yl}benzoic acid 2222117-73-7 详细
4-(3-amino-2,2,4,4-tetramethyl-cyclobutoxy)-2-chloro-benzonitrile;hydrochloride 2891598-69-7 详细
cis-2-phenylcyclopropanamine;hydrochloride 盐酸顺-2-苯基环丙基胺 54779-58-7 详细
tert-butyl 3-piperazin-1-ylazetidine-1-carboxylate 178311-48-3 详细
3-(4-fluorophenyl)oxetan-3-yl]methanol 3-(4-氟苯基)噁丁环烷-3-基]甲醇 1378472-32-2 详细
2-chloro-5-[(2S,3S,4R,5R,6R)-3,4,5-tris(benzyloxy)-6-[(benzyloxy)methyl]oxan-2-yl]benzoic acid 2-氯-5-[(2S,3S,4R,5R,6R)-3,4,5-三(苄氧基)-6-[(苄氧基)甲基]噁烷-2-基]苯甲酸 842133-80-6 详细
5-bromo-2-cyclopropyl-1H-pyrrolo[2,3-b]pyridine 5-溴-2-环丙基-1H-吡咯并[2,3-b]吡啶 1534381-80-0 详细
1-(pyrimidin-2-yl)pyrrolidin-3-amine dihydrochloride 1-(嘧啶-2-基)吡咯烷-3-胺二盐酸 2098048-53-2 详细
trans-2-(4-chloro-3-fluoro-phenyl)cyclopropanecarboxylic acid (1R,2R)-rel-2-(4-氯-3-氟苯基)环丙烷-1-羧酸 2055841-07-9 详细
3-(2-chlorophenoxy)azetidine hydrochloride 1188375-01-0 详细
trans-2-(2-pyridyl)cyclopropanecarboxylic acid 731811-62-4 详细
1-(cyclopropanesulfonyl)azetidin-3-ol 1187594-22-4 详细
hemioxalate 3-(oxetan-3-yl)azetidine 1956369-40-6 详细
2-phenylpyrrolidine 2-苯基吡咯烷 1006-64-0 详细
6-(4-tert-butoxycarbonylpiperazin-1-yl)pyridine-2-carboxylic acid 1175689-45-8 详细
cis-2-phenylsulfanylcyclopropanecarboxylic acid 2135442-61-2 详细
tert-butyl 4-(6-aminopyridin-3-yl)piperazine-1-carboxylate 叔-丁基 4-(6-氨基吡啶-3-基)哌嗪-1-甲酸基酯 571188-59-5 详细
2-chloro-8-cyclopentyl-5-methyl-7H,8H-pyrido[2,3-d]pyrimidin-7-one 2-氯-8-环戊基-5-甲基-7H,8H-吡啶并[2,3-d]嘧啶-7-酮 1013916-37-4 详细
1-[4-(4-amino-3-methoxyphenyl)piperazin-1-yl]ethan-1-one 2-甲氧基-4-(N-乙酰基-哌嗪-1-基)苯胺 1021426-42-5 详细
4-(4-chloro-2-fluorophenyl)-2-methylpyridine-3-carboxylic acid 4-(4-氯-2-氟苯基)-2-甲基吡啶-3-羧酸 1551407-47-6 详细
2-(4-chlorophenyl)imidazo[1,2-a]pyrimidine 56921-86-9 详细
2-hydroxy-N-[(3S)-4-methylene-5-oxo-tetrahydrofuran-3-yl]benzamide 1443448-82-5 详细
methyl cis-3-hydroxy-3-phenyl-cyclobutanecarboxylate 69584-45-8 详细
2-fluoro-3-phenyl-bicyclo[1.1.1]pentane-1-carboxylic acid 2648962-09-6 详细
6-(1-cyanocyclopropyl)imidazo[1,2-a]pyridine-2-carboxylic acid 2654760-79-7 详细
tert-butyl 3-(2-furylmethylsulfonyl)azetidine-1-carboxylate 2940940-70-3 详细
tert-butyl (3R)-cis-4-(4-aminocyclohexyl)-3-(methoxymethyl)piperazine-1-carboxylate 2891580-62-2 详细
3-(4-chlorophenoxy)azetidine;hydrochloride 490021-97-1 详细
5-bromo-1-[[2-fluoro-6-(trifluoromethyl)phenyl]methyl]-6-methylpyrimidine-2,4-dione 5-溴-1-{[2-氟-6-(三氟甲基)苯基]甲基}-6-甲基-1,2,3,4-四氢嘧啶-2,4-二酮 830346-48-0 详细
1-(benzothiophen-4-yl)piperazine;hydrochloride 913614-18-3 详细
ethyl 3-(4-bromophenyl)oxetane-3-carboxylate 1370035-61-2 详细
6-bromo-3-cyclopropoxy-2-methoxypyridine 1243344-95-7 详细
tert-butyl cis-4-[[(1S)-1-phenylethyl]amino]tetrahydrofuran-3-carboxylate 2227197-33-1 详细
tert-butyl 4-(azetidin-3-yloxy)piperidine-1-carboxylate 2229376-64-9 详细
3-(6-bromo-4-methyl-2-pyridyl)tetrahydrofuran-3-ol 2368946-05-6 详细
(5R)-5-[4-(trifluoromethyl)phenyl]morpholin-3-one 1344584-09-3 详细
1-cyclopropylcyclobutanol 89896-69-5 详细
3-(oxetan-3-ylmethyl)azetidine;hydrochloride 2918778-77-3 详细
4-(bromomethyl)-2-[4-(bromomethyl)-2-pyridyl]pyridine 134457-14-0 详细
4-(4-ethyl-1-piperazinyl)-3-fluoro-benzenamine 4-(4-乙基-1-哌嗪基)-3-氟-苯胺 873537-27-0 详细
1-[4-chloro-2-(3-methyl-1H-pyrazol-1-yl)phenyl]-2,2,2-trifluoroethan-1-one 1- [4-氯-2-(3-甲基-1H-吡唑-1-基)苯基] -2,2,2-三氟乙烷-1-酮 1125828-30-9 详细
1-(3-methylazetidin-3-yl)pyrrolidine;dihydrochloride 1152111-80-2 详细
trans-2-phenylcyclopropanamine;hydrochloride 盐酸反-2-苯基环丙基胺 1986-47-6 详细
3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)aniline 641571-11-1 详细
tert-butyl N-[trans-2-(6-bromo-3-pyridyl)cyclopropyl]carbamate 叔-丁基 N-[(1S,2R)-rel-2-(6-溴吡啶-3-基)环丙基]氨基甲酯 918305-73-4 详细
1-[(3,3-difluorocyclobutyl)methyl]-4-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole 1-[(3,3-二氟环丁基)甲基]-4-(四甲基-1,3,2-二噁硼戊环-2-基)-1H-吡唑 2101934-11-4 详细
1-phenylcyclopropane-1-sulfonyl chloride 1-苯基环丙烷-1-磺酰氯化 1359655-41-6 详细
4-(dimethylamino)-4-(3-methoxyphenyl)cyclohexan-1-one 4-(二甲氨基)-4-(3-甲氧苯基)环己烷-1-酮 65618-98-6 详细
4-(morpholine-4-carbonyl)aniline 4-(吗啉-4-羰基)苯胺 51207-86-4 详细
4-ethyl-3-(2-{pyrazolo[1,5-a]pyrimidin-6-yl}ethynyl)benzoic acid 4-乙基-3-(2-{吡唑并[1,5-a]嘧啶-6-基}乙炔基)苯甲酸 1429618-03-0 详细
1-(5-bromopyrimidin-2-yl)cyclobutanol 1515923-39-3 详细
tert-butyl 3-(2,3-difluorophenyl)-3-hydroxyazetidine-1-carboxylate 1227617-37-9 详细
(3S)-3-phenylpiperidine 59349-71-2 详细
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