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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
2-(1,4-diazepan-1-yl)-2-(3-thienyl)acetic acid 1218322-24-7 详细
4-[(6-chloropyrimidin-4-yl)amino]benzoic acid 848639-97-4 详细
3-(4-bromophenyl)-2-azaspiro[3.3]heptane;hydrochloride 2830344-68-6 详细
5-(azetidin-3-yl)-1H-1,2,4-triazole;hydrochloride 2970213-93-3 详细
(3R,5S)-5-(2-pyridyl)pyrrolidin-3-ol;dihydrochloride 2940870-70-0 详细
4-amino-1-[(2R,4R,5R)-5-azido-3,3-difluoro-4-hydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl]pyrimidin-2-one 1145869-51-7 详细
7-[(4-bromophenyl)methyl]-2-oxa-7-azaspiro[3.5]nonane 1200131-53-8 详细
1-(2,4-dichlorophenyl)cyclobutanecarbonitrile 151157-59-4 详细
4-[(3R)-3-piperidyl]benzoic acid 1336552-91-0 详细
(3S)-3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione 57288-03-6 详细
(3S)-3-[4-(trifluoromethyl)phenyl]morpholine 1213924-94-7 详细
N2-methyl-N4-(4-piperidyl)-6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidine-2,4-diamine 2134170-30-0 详细
(2R,3S,4R,5R)-3,4-dihydroxy-5-[(4Z)-4-hydroxyimino-2-oxo-pyrimidin-1-yl]tetrahydrofuran-2-yl]methyl 2-methylpropanoate 2492423-29-5 详细
2-(oxetan-3-yl)pyrazol-3-yl]boronic acid 2304635-25-2 详细
1-[2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazol-1-yl]ethyl]azetidine-3-carbonitrile 1853186-45-4 详细
8-amino-5-bromo-N-cyclopropyl-1,7-naphthyridine-3-carboxamide 2410309-66-7 详细
3-(4-fluorophenyl)bicyclo[1.1.1]pentan-1-amine hydrochloride 2306270-21-1 详细
ethyl 1-[(2-chlorophenyl)methyl]pyrazole-4-carboxylate 1493994-04-9 详细
(3R,4S)-3-cyclopropyl-4-methyl-2-oxo-pyrrolidine-3-carbonitrile 2891580-95-1 详细
1-(4-methylsulfanylpyrimidin-2-yl)pyrrolidin-3-amine;hydrochloride 2940953-33-1 详细
5-methyl-1-phenyl-pyrazole-4-carboxylic acid 91138-00-0 详细
2-anilino-1,2-bis(4-chlorophenyl)ethanone 857561-19-4 详细
trans-2-(4-bromo-3-fluoro-phenyl)cyclopropanamine;hydrochloride 1807941-93-0 详细
3-(1,4-diazepan-1-ylsulfonyl)benzoic acid 1267215-92-8 详细
(1S,2S)-2-(3-fluoro-4-methoxy-phenyl)cyclopropanecarboxylic acid 1609290-18-7 详细
tert-butyl 4-(1H-imidazol-2-ylmethyl)piperazine-1-carboxylate 2891598-88-0 详细
ethyl trans-4-[3-(difluoromethyl)-4-nitro-pyrazol-1-yl]cyclohexanecarboxylate 2750903-83-2 详细
2-trimethylsilylethyl 2-[2-[(1S)-3-(3,4-dimethoxyphenyl)-1-hydroxy-propyl]phenoxy]acetate 2954727-19-4 详细
2-(4-fluorophenyl)indazole 81265-90-9 详细
3-(4-bromophenyl)azetidine 7215-01-2 详细
3-(3-fluorophenoxy)azetidine hydrochloride 1236861-75-8 详细
5-(1,4-diazepan-1-yl)-3-methyl-1,2,4-thiadiazole 1354961-32-2 详细
3-(3-bromophenyl)cyclobutanamine 1156295-97-4 详细
(3R,4R,5R)-2-(4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-3,4-dibenzyloxy-5-(benzyloxymethyl)tetrahydrofuran-2-ol (3R,4R,5R)-2-(4-氨基吡咯并[2,1-f][1,2,4]三嗪-7-基)-3,4-二苄氧基-5-(苄氧基甲基)四氢呋喃丙-2-醇 1355049-94-3 详细
4-amino-1-[(2R,4S,5R)-4-[tert-butyl(dimethyl)silyl]oxy-5-[[tert-butyl(dimethyl)silyl]oxymethyl]tetrahydrofuran-2-yl]-5-(hydroxymethyl)pyrimidin-2-one 1257247-39-4 详细
4-(2-fluorocyclopropyl)phenyl]methanol 1895244-04-8 详细
1-(3-piperazin-1-ylazetidin-1-yl)ethanone;dihydrochloride 2757730-02-0 详细
(3R)-1-cyclopropylpiperidin-3-amine;dihydrochloride 2813579-64-3 详细
N-[(1R)-1-phenylethyl]oxetan-3-amine;hydrochloride 2922439-24-3 详细
methyl (2S)-2-(2-methoxyphenyl)pyrrolidine-3-carboxylate;hydrochloride 2940933-81-1 详细
cis-2-phenylpyrrolidine-3-carboxylic acid hydrochloride 1187927-05-4 详细
2-(2,6-dioxo-3-piperidyl)-5-fluoro-isoindoline-1,3-dione 835616-61-0 详细
N-[(1-methyl-4,5,6,7-tetrahydroindazol-3-yl)methyl]-3-(2-thienyl)prop-2-enamide 1448139-70-5 详细
1-[2-amino-1-(2,5-dimethoxyphenyl)ethyl]pyrrolidine-3-carboxylic acid;dihydrochloride 2940963-65-3 详细
benzyl 4-[5-bromo-6-[(1S)-1-methoxyethyl]-3-pyridyl]piperazine-1-carboxylate 2641451-78-5 详细
2-fluoro-3-methyl-4-([1,2,4]triazolo[1,5-a]pyridin-7-yloxy)aniline 2387518-94-5 详细
3-[[5-[2,2-dimethyl-4-(oxetan-3-yl)piperazin-1-yl]-2-pyridyl]amino]-1-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-one 2696453-81-1 详细
1-(azetidin-3-yl)-N,N-dimethyl-azetidin-3-amine;trihydrochloride 2702323-53-1 详细
(E)-(5-fluoro-3-pyridyl)-(6-fluoro-2-pyridyl)diazene 2387607-48-7 详细
6-bromo-N-cyclopropyl-1H-indole-2-carboxamide 2247646-32-6 详细
2-[2-(adamantane-1-carbonyloxy)-5-oxo-4-oxatricyclo[4.2.1.03]nonane-9-carbonyl]oxy-1,1-difluoro-ethanesulfonate;triphenylsulfonium 2446472-35-9 详细
tert-butyl trans-4-(4-aminocyclohexyl)piperazine-1-carboxylate 876371-20-9 详细
methyl 2-(2-methoxycarbonylphenoxy)carbonyloxybenzoate 82091-12-1 详细
trans-3-(4-fluoro-2-methoxyphenoxy)cyclobutan-1-amine hydrochloride 反-3-(4-氟-2-甲氧基苯氧基)环丁烷-1-胺盐酸 1630906-51-2 详细
(2R,3R,4R,5R)-2-(4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-3,4-dibenzyloxy-5-(benzyloxymethyl)tetrahydrofuran-2-carbonitrile (2R,3R,4R,5R)-2-(4-氨基吡咯并[2,1-f] [1,2,4]三嗪-7-基)-3,4-二苄氧基-5-(苄氧基甲基)四氢呋喃-2-腈 1355357-49-1 详细
tert-butyl 4-[2-(4-chloro-2-fluoro-phenyl)-2-methyl-1,3-benzodioxol-4-yl]piperidine-1-carboxylate 2401894-40-2 详细
4-chloro-2-(6-oxo-2,5-diazatricyclo[7.5.0.02]tetradeca-1(9),7-dien-5-yl)pyridine-3-carbaldehyde 2387601-63-8 详细
1-(1-bicyclo[1.1.1]pentanyl)-4-bromo-pyrazole 2417226-93-6 详细
5-[1-(2-methoxyethyl)pyrazol-4-yl]-2,1,3-benzoxadiazole 2094409-84-2 详细
methyl 2-(6-azaspiro[2.5]octan-6-yl)-4-iodo-benzoate 2600559-83-7 详细
5-[[3-methoxy-4-[(4-nitrophenyl)methoxy]phenyl]methylene]thiazolidine-2,4-dione 331660-78-7 详细
3-(3-chlorophenyl)cyclobutan-1-amine 1156296-61-5 详细
2-pyrrolidin-3-yl-5-(trifluoromethyl)pyridine;dihydrochloride 1909318-71-3 详细
tert-butyl (3S)-3-(1H-pyrazol-3-yl)azepane-1-carboxylate 2380893-98-9 详细
4-[[(1-ethylpyrazolo[3,4-b]pyridin-4-yl)amino]methyl]benzenesulfonamide 2660180-80-1 详细
4-amino-1-[(2R,4S,5R)-4-[tert-butyl(dimethyl)silyl]oxy-5-[[tert-butyl(dimethyl)silyl]oxymethyl]tetrahydrofuran-2-yl]-2-oxo-pyrimidine-5-carboxylic acid 1630012-78-0 详细
tert-butyl 5-(3-methoxycarbonylphenyl)-3,6-dihydro-2H-pyridine-1-carboxylate 2955551-55-8 详细
tert-butyl N-[(3R,4S)-4-phenylpyrrolidin-3-yl]carbamate;hydrochloride 2940858-36-4 详细
methyl (2R)-1-[(1R)-1-phenylethyl]azetidine-2-carboxylate 249734-38-1 详细
4-[(azetidin-3-yl)methyl]morpholine dihydrochloride 1323155-31-2 详细
2-(2,5-difluorophenyl)pyrrolidine 2-(2,5-二氟苯基)吡咯烷 886503-15-7 详细
2-(2,6-dioxo-3-piperidyl)-1-oxo-isoindoline-5-carboxylic acid 2171780-01-9 详细
(3S)-3-(4-bromophenyl)piperidin-2-one 2452378-16-2 详细
2-(1,4-diazepan-1-yl)-2-(2-naphthyl)acetic acid 1218598-47-0 详细
1-[[(3S)-3-fluoropyrrolidin-1-yl]methyl]cyclopropyl]methanol 2708341-87-9 详细
(4-amino-5,6-dimethyl-thieno[2,3-d]pyrimidin-2-yl)methyl 2-amino-4-fluoro-5-methyl-benzoate 2419588-76-2 详细
ethyl trans-2-(4-chloro-3-fluoro-phenyl)cyclopropanecarboxylate 2940858-37-5 详细
trans-2-(1-isobutylpyrazol-4-yl)cyclopropanamine;dihydrochloride 2742942-57-8 详细
1-(4-bromophenyl)-5-methyl-triazol-4-yl]methanol 1239840-96-0 详细
(2R,3R,4S,5R)-2-(6-aminopurin-9-yl)-5-(hydroxymethyl)-4-(2-methoxyethoxy)tetrahydrofuran-3-ol 303197-30-0 详细
3-bromo-2-(4-fluorophenyl)indazole 2281761-79-1 详细
(2S)-2-[2-(propan-2-yl)phenyl]pyrrolidine 1212895-72-1 详细
(3S)-8-Fluoro-1-methyl-3-[2-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-2,4(1H,3H)-quinazolinedione 1643446-65-4 详细
1-methyl-3-[[5-[(2R)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]-2-pyridyl]amino]-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-one 1433849-94-5 详细
1-[2-(2-aminoethoxy)-5-chloro-3-pyridyl]-3-[2-chloro-7-[(1S)-1-methoxyethyl]pyrazolo[1,5-a]pyrimidin-6-yl]urea 2225148-33-2 详细
trans-2-pyrrolidin-1-ylcyclopentanol 32635-39-5 详细
N-(4-bromo-2,5-difluoro-phenyl)-6-chloro-1H-pyrrolo[2,3-b]pyridine-3-sulfonamide 2231232-39-4 详细
(2'R,4'S)-9'-[(2'R,4'S)-2,2-dimethylspiro[1,3-dioxane-5,3'-10-azatricyclo[4.4.0.02]deca-1(6),7,9-triene]-9'-yl]-2,2-dimethyl-spiro[1,3-dioxane-5,3'-10-azatricyclo[4.4.0.02]deca-1(6),7,9-triene 2761045-11-6 详细
(3S)-6-(5-ethyl-1,2,4-oxadiazol-3-yl)-2,3-dihydrobenzofuran-3-amine;hydrochloride 2364560-92-7 详细
trans-2,2-dimethyl-3-phenyl-cyclopropanamine;hydrochloride 2940870-52-8 详细
3-(4-fluorophenyl)-1H-pyrimidine-2,4-dione 1204297-90-4 详细
cis-3-[4-(trifluoromethyl)phenyl]cyclobutanamine 1812174-93-8 详细
4-morpholin-2-ylphenol;hydrochloride 103030-79-1 详细
3-(4-chloropyrimidin-2-yl)-1-methyl-indole 2364486-23-5 详细
tert-butyl 4-(4-methoxycarbonyl-1-bicyclo[2.2.2]octanyl)piperazine-1-carboxylate 2891599-76-9 详细
trans-5-(2-pyridyl)pyrrolidin-3-ol;dihydrochloride 2940872-22-8 详细
8-chloro-4-(dimethylaminomethylene)-1-(2-fluoro-6-methoxy-phenyl)-3H-2-benzazepin-5-one 869367-33-9 详细
4-[(2S)-pyrrolidin-2-yl]benzoic acid 1213448-39-5 详细
(4-bromophenyl)(cyclopropyl)methanone 6952-89-2 详细
3-(4-bromo-3-methyl-2-oxo-benzimidazol-1-yl)piperidine-2,6-dione 2304754-51-4 详细
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