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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
5-methyl-2-(pyrimidin-2-yl)benzoic acid 1088994-22-2 详细
4-chloro-7-methylpyrido[2,3-d]pyrimidine 4-氯-7-甲基吡啶并[2,3-d]嘧啶 117890-81-0 详细
(2S,3R)-3-phenylpyrrolidine-2-carboxylic acid 118758-48-8 详细
2-cyclopropylpyrimidin-5-amine 2-环丙基嘧啶-5-胺 1152519-69-1 详细
CNX-774 1202759-32-7 详细
Zamicastat 1080028-80-3 详细
(+)-Tetrabenazine (+)-丁苯那嗪; (3R,11bR)-1,3,4,6,7,11b-六氢-9,10-二甲氧基-3-异丁基-2H-苯并[a]喹嗪-2-酮 1026016-83-0 详细
tert-butyl N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)carbamate 1158767-01-1 详细
4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridine-2-carboxylic acid hydrochloride 4H,5H,6H,7H-[1,3]噻唑并[5,4-c]吡啶-2-羧酸盐酸 1190971-73-3 详细
GDC-0425 1200129-48-1 详细
2-fluoro-5-methoxy-4-nitro-benzoic acid 1001345-80-7 详细
tert-butyl 5'-bromo-2'-oxo-1',2'-dihydrospiro[piperidine-4,3'-pyrrolo[2,3-b]pyridine]-1-carboxylate 叔-丁基 5'-溴-2'-氧亚基-1',2'-二氢螺[哌啶并-4,3'-吡咯并[2,3-b]吡啶]-1-甲酸基酯 1192834-16-4 详细
(S)-methyl 4-oxo-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxylate 1190392-23-4 详细
2-[(2-carboxyphenyl)disulfanyl]benzoic acid 119-80-2 详细
6'-bromo-1',2'-dihydrospiro[oxane-4,3'-pyrrolo[3,2-b]pyridine]-2'-one 1190862-19-1 详细
6-methoxy-1,2,3,4-tetrahydroquinoline 120-15-0 详细
4,4-dimethyl-6,7-dihydro-5H-thieno[3,2-c]pyridine 1176404-23-1 详细
tricyclo[9.4.0.03]pentadeca-1(11),3(8),4,6,9,12,14-heptaen-2-one oxime 1021-91-6 详细
5H,6H,7H-cyclopenta[b]pyridin-5-ol 1065609-70-2 详细
3-(7-bromo-2-methyl-4-oxo-quinazolin-3-yl)piperidine-2,6-dione 1135008-81-9 详细
ditert-butyl-[3,6-dimethoxy-2-(2,4,6-triisopropylphenyl)phenyl]phosphane 1160861-53-9 详细
(2S)-3-[tert-butoxycarbonyl(isopropyl)amino]-2-(4-chlorophenyl)propanoic acid 1001179-33-4 详细
tert-butyl 4-(4-bromo-5-methyl-pyrazol-1-yl)piperidine-1-carboxylate 1076223-99-8 详细
3-(benzenesulfonyl)propanoic acid 10154-71-9 详细
tert-butyl 2-chloro-5H,6H,7H,8H-pyrido[4,3-d]pyrimidine-6-carboxylate 2-氯-7,8-二氢吡啶并[4,3-D]嘧啶-6(5H)-甲酸叔丁酯 1092352-55-0 详细
Gedatolisib 1197160-78-3 详细
1-[2-(4-methylpiperazin-1-yl)ethyl]-1H-pyrazol-4-amine 1201363-83-8 详细
{2H-[1,3]dioxolo[4,5-b]pyridin-6-yl}boronic acid 1019767-68-0 详细
1h-benzimidazole, 2-[[[4-(3-methoxypropoxy)-3-methyl-2-pyridinyl]methyl]sulfinyl]- 117976-89-3 详细
chromane-3-carboxylic acid 115822-57-6 详细
2-chloro-6-(3-methoxyphenyl)pyrimidine-4-carboxylic acid 1181712-25-3 详细
4-bromo-1-cyclopropyl-1H-pyrazole 1151802-23-1 详细
3-methoxy-1,5-naphthyridine-4-carbaldehyde 1056877-13-4 详细
(S)-cyclopropyl-(4-fluorophenyl)methanamine hydrochloride 1202478-48-5 详细
Brigatinib 1197953-54-0 详细
methyl 2-methyl-1,2,3,4-tetrahydroisoquinoline-7-carboxylate 1038549-50-6 详细
PRI 2201dene]-4-methylene-cyclohexane-1,3-diol 112965-21-6 详细
3-(5-bromo-1-oxo-isoindolin-2-yl)piperidine-2,6-dione 1010100-26-1 详细
trans-2-(4-cyanophenyl)cyclopropanecarboxylic acid 1119807-15-6 详细
6-bromo-1,2-dihydropyrido[2,3-b][1,4]oxazin-3-one 105544-36-3 详细
2-chloro-6,7-dihydro-5H-cyclopenta[b]pyridine 117890-55-8 详细
Apabetalone 1044870-39-4 详细
Ponatinib hydrochloride 1114544-31-8 详细
Cariprazine hydrochloride 1083076-69-0 详细
jnj39758979 1046447-90-8 详细
tert-butyl (3S)-3-[(5-amino-2-pyridyl)oxy]pyrrolidine-1-carboxylate 1141488-38-1 详细
6-(trifluoromethyl)-2,3-dihydrofuro[2,3-b]pyridin-3-amine 1196156-88-3 详细
3-cyclopropyl-1h-pyrazole 100114-57-6 详细
tert-butyl 3-oxo-5,6,8,9-tetrahydro-2H-pyridazino[3,4-d]azepine-7-carboxylate 1190897-27-8 详细
4-(piperidin-4-yl)aniline 4-(哌啶-4-基)苯胺 113310-52-4 详细
(3-phenyloxetan-3-yl)methanol (3-苯基噁丁环烷-3-基)甲醇 114012-43-0 详细
Alisertib 1028486-01-2 详细
6-tert-butyl 2-ethyl 4H,5H,6H,7H-thieno[2,3-c]pyridine-2,6-dicarboxylate 6-叔-丁基 2-乙基 4H,5H,6H,7H-噻吩并[2,3-c]吡啶-2,6-二甲酸基酯 1135124-02-5 详细
(2S)-2-amino-2-(m-tolyl)ethanol 1026230-99-8 详细
(2-chloro-5-formylphenyl)boronic acid 1150114-78-5 详细
4-phenylpyrrolidin-2-one 4-苯基吡咯烷-2-酮 1198-97-6 详细
5,6,7,8-tetrahydro-2H-cyclohepta[c]pyrrol-4-one 113880-81-2 详细
2-bromo-4H,5H,6H,7H-thieno[3,2-c]pyridin-4-one 2-溴-4H,5H,6H,7H-噻吩并[3,2-c]吡啶-4-酮 1078150-17-0 详细
1-cyclopropylpyrazole-4-carbaldehyde 1082066-00-9 详细
1-methyl-5,6-dihydro-4H-pyrrolo[3,4-c]pyrazole;hydrochloride 1187830-68-7 详细
1-pyrazin-2-ylcyclopropanecarbonitrile 1159734-50-5 详细
finerenone 1050477-31-0 详细
tert-butyl 2-amino-4-(4-methylpiperazin-1-yl)benzoate 1034975-35-3 详细
Valbenazine 卫本呐嗪;(2R,3R,11bR)-9,10-二甲氧基-3-(2-甲基丙基)-1H,2H,3H,4H,6H,7H,11bH-吡啶[2,1-a]异喹啉-2-取代,(2S)-2-氨基-3-甲基丁酸酯 1025504-45-3 详细
(3S)-6-fluoro-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid 1161833-81-3 详细
(5-chloro-3-pyridyl) 1H-indole-5-carboxylate 1026559-41-0 详细
3-bromobicyclo[4.2.0]octa-1,3,5-triene 1073-39-8 详细
(3R)-2,3,4,9-tetrahydro-1H-carbazol-3-amine 116650-33-0 详细
4-bromo-2-fluoro-1-iodobenzene 4-溴-2-氟-1-碘苯 105931-73-5 详细
2-fluoro-3-hydroxybenzaldehyde 103438-86-4 详细
Niraparib 2-[4-((3S)-3-哌啶基)苯基]-2H-吲唑-7-甲酰胺 1038915-60-4 详细
Evacetrapib 1186486-62-3 详细
4-bromo-7-fluoro-indan-1-one 1003048-72-3 详细
Baricitinib 1187594-09-7 详细
2-chloro-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenol 1151564-17-8 详细
(3,5-difluoro-4-methoxycarbonyl-phenyl)boronic acid 1190989-09-3 详细
7-phenyl-7-(2,4,5-trimethyl-3,6-dioxocyclohexa-1,4-dien-1-yl)heptanoic acid 112665-43-7 详细
5,6,7,8-tetrahydroquinoline-2-carbaldehyde 1071063-42-7 详细
cis-1-tert-butoxycarbonyl-3-phenyl-piperidine-4-carboxylic acid 1068522-21-3 详细
4-(1-methylpyrazol-4-yl)piperidine 1138218-02-6 详细
methyl 6-oxo-4,5-dihydro-1H-cyclopenta[b]pyrrole-2-carboxylate 1041430-92-5 详细
7-morpholino-6,7,8,9-tetrahydro-5H-benzo[7]annulen-3-amine 1022963-80-9 详细
2H,4H,5H,6H,7H,7aH-thieno[3,2-c]pyridin-2-one 2H,4H,5H,6H,7H,7aH-噻吩并[3,2-c]吡啶-2-酮 109904-37-2 详细
ethyl 2-amino-4-cyclopropyl-thiophene-3-carboxylate 120109-75-3 详细
2-chloro-6-cyclopropylpyridine-3-carbonitrile 1198475-35-2 详细
Telotristat ethyl 泰乐曲丝坦 1033805-22-9 详细
1,2,5,6,7,8-hexahydro-2,6-naphthyridin-1-one 1170830-85-9 详细
1-(1-methylpiperidin-4-yl)-1h-pyrazol-4-amine 1-(1-甲基哌啶-4-基)-1h-吡唑-4-胺 1201935-36-5 详细
5-bromo-2-[3-(chloromethyl)phenyl]pyrimidine 5-溴-2-[3-(氯甲基)苯基]嘧啶 1100598-50-2 详细
CORT-108297 1018679-79-2 详细
Lifitegrast 1025967-78-5 详细
2-(2-chlorophenyl)cyclopropane-1-carboxylic acid 2-(2-氯苯基)环丙烷-1-羧酸 1181230-38-5 详细
Letrozole 112809-51-5 详细
2,4-dichloro-7,8-dihydro-6H-quinolin-5-one 1028330-50-8 详细
3-chloro-4-imidazo[1,2-a]pyridin-7-yloxy-aniline 1033810-67-1 详细
(1S,4R,7R,9S,10S,13R,15S)-15-hydroxy-7-[(2R,3R,4R,5R,6R)-6-(hydroxymethyl)-3-(3-methylbutanoyloxy)-4,5-disulfooxy-tetrahydropyran-2-yl]oxy-9-methyl-14-methylene-tetracyclo[11.2.1.011o.0]hexadecane-5-carboxylic acid;bis(potassium salt) 102130-43-8 详细
5-(p-tolyl)-2H-1,2,4-triazin-3-one 1199767-11-7 详细
(4S)-3,4-dihydro-2H-1-benzopyran-4-amine hydrochloride 1035093-81-2 详细
methyl 5,5-difluoro-4-oxo-1,6-dihydrocyclopenta[b]pyrrole-2-carboxylate 1041430-63-0 详细
dibenzothiophene 5-oxide 1013-23-6 详细
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