中文名:LY-294,002盐酸盐
英文名:LY-294,002 hydrochloride
纯度:≥98%(HPLC)
货号:L171289
Cas号:934389-88-5
存储温度:-20°C储存
运输条件:超低温运输
产品介绍:
Product Describtion:
LY-294,002 hydrochloride is a derivative of the flavonoid, quercetin and elicits higher inhibition on the enzyme phosphoinositide 3-kinase (PI3K). LY-294,002 inhibits nuclear factor kappa B signaling in macrophages. It elevates expression of autophagosomal protein LC3 and promotes apoptosis in gastric and nasopharyngeal cancer cells. LY-294,002 modulates action potential repolarization and improves myocyte contractility.
Product Application:
LY-294,002 hydrochloride has been used in the inhibition of:
phosphoinositide 3-kinase (PI3K) in human lung cancer cell line
autophagy in mesenchymal stem cells (MSCs).
serine/threonine-specific protein kinase (AKT) signaling in fibroblasts and cardiac cells.
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关键字: 2-(4-吗啉基)-8-苯基-1(4H)-苯并吡喃-4-酮 盐酸盐;EX-A1710 ; 2-morpholin-4-yl-8-phenylchromen-4-one,hydrochloride ; AS-58350
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