Bretazenil
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- $41 - $2500
- Product name: Bretazenil
- CAS: 84379-13-5
- MF: C19H20BrN3O3
- MW: 418.28
- EINECS:240-723-0
- MDL Number:MFCD00866987
- Synonyms:9H-IMIDAZO(1,5-A)PYRROLO(2,1-C)(1,4)BENZODIAZEPINE-1-CARBOXYLIC ACID,11,12,13,13A-TTRRRAHYDRO-8-BROMO-9-OXO-,1,1-DIMETHYLETHYL ESTER,(S)-;1,1-dimethylethylester,(s)-13a-tetrahydro-8-bromo-9-oxo ;9h-imidazo(1,5-a)pyrrolo(2,1-c)(1,4)benzodiazepine-1-carboxylicacid,11,12,13, ;(13aS)-8-Bromo-9-oxo-11,12,13,13a-tetrahydro-9H-imidazo[1,5-a]pyrrolo[2,1-c][1,4]benzodiazepine-1-carboxylic acid tert-butyl ester;9H-Imidazo(1,5-A)pyrrolo(2,1-C)(1,4)benzodiazepine-1-carboxylic acid, 8-bromo-11,12,13,13A-tetrahydro-9-oxo-, 1,1-dimethylethyl ester, (S)-;Bretazenilum;Bretazenilum [inn-latin];Brn 4765855
34 prices
Selected condition：
Brand
- aablocks
- AK Scientific
- ApexBio Technology
- Biorbyt Ltd
- Biosynth
- Cayman Chemical
- ChemScene
- DC Chemicals
- Labseeker
- Sigma-Aldrich
- Usbiological
Package
- 1mg
- 5mg
- 10mg
- 25mg
- 50mg
- 100mg
- 250mg
- 500mg
- Manufactureraablocks
- Product numberAA00G600
- Product descriptionBretazenil 40mgin1mLDMSO
- Packaging5mg
- Price$125
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00G600
- Product descriptionBretazenil 40mgin1mLDMSO
- Packaging10mg
- Price$180
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00G600
- Product descriptionBretazenil 40mgin1mLDMSO
- Packaging25mg
- Price$331
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00G600
- Product descriptionBretazenil 40mgin1mLDMSO
- Packaging50mg
- Price$533
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00G600
- Product descriptionBretazenil 40mgin1mLDMSO
- Packaging100mg
- Price$889
- Updated2026-05-28
- Buy
- ManufacturerAK Scientific
- Product number7816CA
- Product descriptionBretazenil
- Packaging10mg
- Price$256
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product number7816CA
- Product descriptionBretazenil
- Packaging25mg
- Price$442
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB7430
- Product descriptionBretazenil
- Packaging25mg
- Price$350
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberB7430
- Product descriptionBretazenil
- Packaging10mg
- Price$170
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberB7430
- Product descriptionBretazenil
- Packaging5mg
- Price$100
- Updated2026-05-06
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb1473105
- Product descriptionRo 16-6028 >98%
- Packaging100mg
- Price$520
- Updated2026-05-06
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb1473105
- Product descriptionRo 16-6028 >98%
- Packaging250mg
- Price$890
- Updated2026-05-06
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb1473105
- Product descriptionRo 16-6028 >98%
- Packaging500mg
- Price$1630
- Updated2026-05-06
- Buy
- ManufacturerBiosynth
- Product numberJDA37913
- Product descriptionBretazenil
- Packaging100mg
- Price$2500
- Updated2026-06-04
- Buy
- ManufacturerBiosynth
- Product numberJDA37913
- Product descriptionBretazenil
- Packaging50mg
- Price$1562.5
- Updated2026-06-04
- Buy
- ManufacturerBiosynth
- Product numberJDA37913
- Product descriptionBretazenil
- Packaging25mg
- Price$1123.5
- Updated2026-06-04
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA00G600 | Bretazenil 40mgin1mLDMSO | 5mg | $125 | 2026-05-28 | Buy |
| aablocks | AA00G600 | Bretazenil 40mgin1mLDMSO | 10mg | $180 | 2026-05-28 | Buy |
| aablocks | AA00G600 | Bretazenil 40mgin1mLDMSO | 25mg | $331 | 2026-05-28 | Buy |
| aablocks | AA00G600 | Bretazenil 40mgin1mLDMSO | 50mg | $533 | 2026-05-28 | Buy |
| aablocks | AA00G600 | Bretazenil 40mgin1mLDMSO | 100mg | $889 | 2026-05-28 | Buy |
| AK Scientific | 7816CA | Bretazenil | 10mg | $256 | 2021-12-16 | Buy |
| AK Scientific | 7816CA | Bretazenil | 25mg | $442 | 2021-12-16 | Buy |
| ApexBio Technology | B7430 | Bretazenil | 25mg | $350 | 2026-05-06 | Buy |
| ApexBio Technology | B7430 | Bretazenil | 10mg | $170 | 2026-05-06 | Buy |
| ApexBio Technology | B7430 | Bretazenil | 5mg | $100 | 2026-05-06 | Buy |
| Biorbyt Ltd | orb1473105 | Ro 16-6028 >98% | 100mg | $520 | 2026-05-06 | Buy |
| Biorbyt Ltd | orb1473105 | Ro 16-6028 >98% | 250mg | $890 | 2026-05-06 | Buy |
| Biorbyt Ltd | orb1473105 | Ro 16-6028 >98% | 500mg | $1630 | 2026-05-06 | Buy |
| Biosynth | JDA37913 | Bretazenil | 100mg | $2500 | 2026-06-04 | Buy |
| Biosynth | JDA37913 | Bretazenil | 50mg | $1562.5 | 2026-06-04 | Buy |
| Biosynth | JDA37913 | Bretazenil | 25mg | $1123.5 | 2026-06-04 | Buy |
Properties
Boiling point :594.3±50.0 °C(Predicted)
Density :1.56±0.1 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO: 24 mg/mL, soluble
form :solid
pka :0.78±0.20(Predicted)
color :white
InChI :InChI=1S/C19H20BrN3O3/c1-19(2,3)26-18(25)15-16-13-8-5-9-22(13)17(24)14-11(20)6-4-7-12(14)23(16)10-21-15/h4,6-7,10,13H,5,8-9H2,1-3H3/t13-/m0/s1
InChIKey :LWUDDYHYYNNIQI-ZDUSSCGKSA-N
SMILES :N12C=NC(C(OC(C)(C)C)=O)=C1[C@]1([H])CCCN1C(=O)C1=C(Br)C=CC=C12
Density :1.56±0.1 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO: 24 mg/mL, soluble
form :solid
pka :0.78±0.20(Predicted)
color :white
InChI :InChI=1S/C19H20BrN3O3/c1-19(2,3)26-18(25)15-16-13-8-5-9-22(13)17(24)14-11(20)6-4-7-12(14)23(16)10-21-15/h4,6-7,10,13H,5,8-9H2,1-3H3/t13-/m0/s1
InChIKey :LWUDDYHYYNNIQI-ZDUSSCGKSA-N
SMILES :N12C=NC(C(OC(C)(C)C)=O)=C1[C@]1([H])CCCN1C(=O)C1=C(Br)C=CC=C12
Safety Information
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Description
Bretazenil, an imidazobenzodiazepinone, is the first partial benzodiazepine agonist to be evaluated in schizophrenia. Bretazenil has been used to determine non-specific binding due to its affinity to bind to a variety of γ-aminobutyric acid type A (GABAA) receptor subtypes (α1-3;5). It has also been used as a GABAA receptor partial agonist in the subcutaneous Alzet minipumps to treat obese agouti related protein (AgRP) ablated and lean naive mice to study its effect on them.More related product prices
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