-Conotoxin GVIA (trifluoroacetate salt)
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- $602
- Product name: -Conotoxin GVIA (trifluoroacetate salt)
- CAS:
- MF: C122H183F3N38O45S6
- MW: 3151.3712296
- EINECS:
- MDL Number:
- Synonyms:-Conotoxin GVIA (trifluoroacetate salt)
1 prices
Selected condition：
Brand
- Cayman Chemical
Package
- 1mg
- ManufacturerCayman Chemical
- Product number24114
- Product descriptionω-Conotoxin GVIA (trifluoroacetate salt) ≥95%
- Packaging1mg
- Price$602
- Updated2026-04-30
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| Cayman Chemical | 24114 | ω-Conotoxin GVIA (trifluoroacetate salt) ≥95% | 1mg | $602 | 2026-04-30 | Buy |
Properties
solubility :Water: 1 mg/ml
Safety Information
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Description
ω-Conotoxin GVIA is a peptide originally isolated from the marine mollusk C. geographus that acts as an N-type calcium channel blocker.1,2 It binds to human neocortical, rat hippocampal, and chick brain synaptic plasma membranes (IC50s = 4.6, 60, and 150 pM, respectively, in radioligand binding assays).3,4,5 ω-Conotoxin GVIA inhibits norepinephrine (Item No. 16673) and acetylcholine (Item No. 23829) release from human neocortical slices (IC50s = 14 and 3 nM, respectively) and calcium influx into chick synaptosomes by 92% when used at a concentration of 0.1 μM.3,4 It blocks electrically-evoked twitch responses of rat vas deferens and guinea pig ileum (IC50s = 9.8 and 55 nM, respectively) but does not affect the postjunctional contractile responses induced by norepinephrine on vas deferens or by carbamoylcholine (carbachol; Item No. 14486) on ileum.6 ω-Conotoxin GVIA does not affect potassium-induced contraction of rat aorta at concentrations up to 1 μM.WARNING This product is not for human or veterinary use.More related product prices