Lapatinib
|
- $10 - $1900
- Product name: Lapatinib
- CAS: 231277-92-2
- MF: C29H26ClFN4O4S
- MW: 581.06
- EINECS:1806241-263-5
- MDL Number:MFCD09264194
- Synonyms:lapatinib;n-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[(2-methylsulfonylethylamino)methyl]-2-furyl]quinazolin-4-amine;4-Quinazolinamine, N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-;Lapatinib(TINIBS);Lapatinib Base N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-Quinazolinamine;GW2016 LAPATINIB;N-(3-chloro-4-((3-fluorobenzyl)oxy)phenyl)-6-(5-(((2-(methylsulfonyl)ethyl)amino)methyl)furan-2-yl)quinazolin-4-amine;N-{3-chloro-4-[(3-fluorobenzyl)oxyl]phenyl}-6-[5-({[2-(methylsulfonyl)ethyl]amino}methyl)furan-2-yl]quinazolin-4-amine
113 prices
Selected condition：
Brand
- aablocks
- AccelPharmtech
- ACHEMBLOCK
- Adipogen Life Sciences
- AK Scientific
- Ambeed
- American Custom Chemicals Corporation
- ApexBio Technology
- Arctom
- AvaChem
- Biorbyt Ltd
- Biosynth
- Cayman Chemical
- ChemScene
- DC Chemicals
- Matrix Scientific
- Medical Isotopes, Inc.
- Sigma-Aldrich
- TCI Chemical
- Thermo Scientific Chemicals
- Tocris
- TRC
- Usbiological
Package
- 5mg
- 10mM*1mLinDMSO(Solid+Solvent)
- 10mM(in 1mL DMSO)
- 10mM(in1mLDMSO)
- 10mg
- 10mM*1mLinDMSO(Solution)
- 10
- 20mg
- 10mM*1mLinDMSO
- 1mg
- 10mM(1mLinDMSO)
- EvaluationSample
- 25mg
- 50mg
- 100mg
- 200mg
- 250mg
- 250.00mg
- 500mg
- 1.00g
- 1000mg
- 1g
- 2g
- 2000mg
- 5.00g
- 5000mg
- 5g
- 10G
- 10000mg
- 25g
- 1 g
- 10 mg
- 50 mg
- Manufactureraablocks
- Product numberAA0039I1
- Product descriptionN-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine 98%
- Packaging1mg
- Price$10
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0039I1
- Product descriptionN-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine ≥99%
- Packaging25mg
- Price$12
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0039I1
- Product descriptionN-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine 99%
- Packaging250mg
- Price$26
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0039I1
- Product descriptionN-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine 98%
- Packaging1g
- Price$49
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0039I1
- Product descriptionN-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine 98%
- Packaging5g
- Price$119
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0039I1
- Product descriptionN-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine 98%
- Packaging25g
- Price$540
- Updated2026-05-28
- Buy
- ManufacturerAccelPharmtech
- Product numberAT7855
- Product descriptionLapatinib 99.00%
- Packaging10G
- Price$240
- Updated2026-05-21
- Buy
- ManufacturerAccelPharmtech
- Product numberAT7855
- Product descriptionLapatinib 99.00%
- Packaging25G
- Price$380
- Updated2026-05-21
- Buy
- ManufacturerAccelPharmtech
- Product numberAT7855
- Product descriptionLapatinib 99.00%
- Packaging5G
- Price$170
- Updated2026-05-21
- Buy
- ManufacturerACHEMBLOCK
- Product number10344
- Product descriptionLapatinib 98%
- Packaging5G
- Price$180
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product number10344
- Product descriptionLapatinib 98%
- Packaging1G
- Price$55
- Updated2026-05-27
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberSYN-1052-M005
- Product descriptionLapatinib ≥95%
- Packaging5mg
- Price$65
- Updated2026-05-06
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberSYN-1052-M001
- Product descriptionLapatinib ≥95%
- Packaging1mg
- Price$54
- Updated2026-05-06
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberSYN-1052-M050
- Product descriptionLapatinib ≥95%
- Packaging50mg
- Price$205
- Updated2026-05-06
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberSYN-1052-M010
- Product descriptionLapatinib ≥95%
- Packaging10mg
- Price$76
- Updated2026-05-06
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberSYN-1052-M100
- Product descriptionLapatinib ≥95%
- Packaging100mg
- Price$292
- Updated2026-05-06
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA0039I1 | N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine 98% | 1mg | $10 | 2026-05-28 | Buy |
| aablocks | AA0039I1 | N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine ≥99% | 25mg | $12 | 2026-05-28 | Buy |
| aablocks | AA0039I1 | N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine 99% | 250mg | $26 | 2026-05-28 | Buy |
| aablocks | AA0039I1 | N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine 98% | 1g | $49 | 2026-05-28 | Buy |
| aablocks | AA0039I1 | N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine 98% | 5g | $119 | 2026-05-28 | Buy |
| aablocks | AA0039I1 | N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine 98% | 25g | $540 | 2026-05-28 | Buy |
| AccelPharmtech | AT7855 | Lapatinib 99.00% | 10G | $240 | 2026-05-21 | Buy |
| AccelPharmtech | AT7855 | Lapatinib 99.00% | 25G | $380 | 2026-05-21 | Buy |
| AccelPharmtech | AT7855 | Lapatinib 99.00% | 5G | $170 | 2026-05-21 | Buy |
| ACHEMBLOCK | 10344 | Lapatinib 98% | 5G | $180 | 2026-05-27 | Buy |
| ACHEMBLOCK | 10344 | Lapatinib 98% | 1G | $55 | 2026-05-27 | Buy |
| Adipogen Life Sciences | SYN-1052-M005 | Lapatinib ≥95% | 5mg | $65 | 2026-05-06 | Buy |
| Adipogen Life Sciences | SYN-1052-M001 | Lapatinib ≥95% | 1mg | $54 | 2026-05-06 | Buy |
| Adipogen Life Sciences | SYN-1052-M050 | Lapatinib ≥95% | 50mg | $205 | 2026-05-06 | Buy |
| Adipogen Life Sciences | SYN-1052-M010 | Lapatinib ≥95% | 10mg | $76 | 2026-05-06 | Buy |
| Adipogen Life Sciences | SYN-1052-M100 | Lapatinib ≥95% | 100mg | $292 | 2026-05-06 | Buy |
Properties
Melting point :144-146oC
Boiling point :750.7±60.0 °C(Predicted)
Density :1.381±0.06 g/cm3(Predicted)
storage temp. :2-8°C(protect from light)
solubility :Soluble in DMSO (up to 200 mg/ml)
pka :6.34±0.19(Predicted)
form :solid
color :Yellow
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
InChIKey :BCFGMOOMADDAQU-UHFFFAOYSA-N
SMILES :N1=C2C(C=C(C3=CC=C(CNCCS(C)(=O)=O)O3)C=C2)=C(NC2=CC=C(OCC3=CC=CC(F)=C3)C(Cl)=C2)N=C1
CAS DataBase Reference :231277-92-2(CAS DataBase Reference)
Boiling point :750.7±60.0 °C(Predicted)
Density :1.381±0.06 g/cm3(Predicted)
storage temp. :2-8°C(protect from light)
solubility :Soluble in DMSO (up to 200 mg/ml)
pka :6.34±0.19(Predicted)
form :solid
color :Yellow
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
InChIKey :BCFGMOOMADDAQU-UHFFFAOYSA-N
SMILES :N1=C2C(C=C(C3=CC=C(CNCCS(C)(=O)=O)O3)C=C2)=C(NC2=CC=C(OCC3=CC=CC(F)=C3)C(Cl)=C2)N=C1
CAS DataBase Reference :231277-92-2(CAS DataBase Reference)
Safety Information
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| Signal word: | Warning | ||||||||||||||||||||||||||||
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Description
The epidermal growth factor (EGF) receptors EGFR (ErbB1) and human EGFR2 (HER2, ErbB2) are receptor tyrosine kinases that are often over-expressed in cancer. Lapatinib is a potent and selective dual inhibitor of EGFR and HER2 (IC50s = 19 and 3 nM, respectively). It is effective in vivo and is used in combination therapy to prevent or suppress cancers where these kinases are over-expressed, including breast cancer.Related product price
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Suppliers and manufacturers
SHANDONG BOYUAN PHARMACEUTICAL CO., LTD.
Lapatinib
CAS:231277-92-2
Hangzhou Hyper Chemicals Limited
Lapatinib
CAS:231277-92-2
BEIJING SJAR TECHNOLOGY DEVELOPMENT CO., LTD.
Capot Chemical Co.,Ltd.
Henan Tianfu Chemical Co.,Ltd.
Jinan Jianfeng Chemical Co., Ltd
Xiamen AmoyChem Co., Ltd
CONIER CHEM AND PHARMA LIMITED
SIMAGCHEM CORP
Lapatinib
CAS:231277-92-2
