(R)-Methyl 4-(2-(3,4-dichlorophenyl)acetyl)-3-(pyrrolidin-1-ylmethyl)piperazine-1-carboxylate fumarate
- CAS No.
- 126766-43-6
- Chemical Name:
- (R)-Methyl 4-(2-(3,4-dichlorophenyl)acetyl)-3-(pyrrolidin-1-ylmethyl)piperazine-1-carboxylate fumarate
- Synonyms
- GR-103545 fumarate;GR103545, 10 mM in DMSO;(R)-(-)-GR103545 fumarate;Inhibitor,Opioid Receptor,imaging,GR103545,inhibit,κ-OR,GR 103545,κ-opioid receptor,GR-103545;(R)-Methyl 4-(2-(3,4-dichlorophenyl)acetyl)-3-(pyrrolidin-1-ylmethyl)piperazine-1-carboxylate fumarate;1-Piperazinecarboxylic acid,4-[(3,4-dichlorophenyl)acetyl]-3-(1- pyrrolidinylmethyl)-,methyl ester,(3R)-,(2E)-2-butenedioate (1:1)
- CBNumber:
- CB19972356
- Molecular Formula:
- C23H29Cl2N3O7
- Molecular Weight:
- 530.4
- MDL Number:
- MFCD00902108
- MOL File:
- 126766-43-6.mol
- MSDS File:
- SDS
(R)-Methyl 4-(2-(3,4-dichlorophenyl)acetyl)-3-(pyrrolidin-1-ylmethyl)piperazine-1-carboxylate fumarate price
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| ChemScene | CS-0356525 | GR103545 | 126766-43-6 | 1mg | $233 | 2026-06-04 | Buy |
| ChemScene | CS-0356525 | GR103545 | 126766-43-6 | 2mg | $375 | 2026-06-04 | Buy |
| ChemScene | CS-0356525 | GR103545 | 126766-43-6 | 5mg | $538 | 2026-06-04 | Buy |
| ChemScene | CS-0356525 | GR103545 | 126766-43-6 | 10mg | $768 | 2026-06-04 | Buy |
| ChemScene | CS-0356525 | GR103545 | 126766-43-6 | 25mg | $1289 | 2026-06-04 | Buy |
(R)-Methyl 4-(2-(3,4-dichlorophenyl)acetyl)-3-(pyrrolidin-1-ylmethyl)piperazine-1-carboxylate fumarate Chemical Properties, Uses, Production
Description
GR-103545 is a reference and non-radio labeled agent. The radio-labeled 11C-GR103545 is a promising PET radiotracer for imaging the κ-OR.
Uses
GR103545 is a potent and selective agonist of the κ-opioid receptor (κ-OR). 11GR103545 is a radiotracer for imaging κ-OR in vivo[1][2].
References
[1] Hayes AG, et, al. A series of novel, highly potent and selective agonists for the kappa-opioid receptor. Br J Pharmacol. 1990 Dec;101(4):944-8. DOI:10.1111/j.1476-5381.1990.tb14185.x
[2] Talbot PS, et, al. 11C-GR103545, a radiotracer for imaging kappa-opioid receptors in vivo with PET: synthesis and evaluation in baboons. J Nucl Med. 2005 Mar;46(3):484-94. PMID:15750163
(R)-Methyl 4-(2-(3,4-dichlorophenyl)acetyl)-3-(pyrrolidin-1-ylmethyl)piperazine-1-carboxylate fumarate Preparation Products And Raw materials
Raw materials
Preparation Products
(R)-Methyl 4-(2-(3,4-dichlorophenyl)acetyl)-3-(pyrrolidin-1-ylmethyl)piperazine-1-carboxylate fumarate Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
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| BOC Sciences | 1-631-485-4226; 16314854226 | info@bocsci.com | United States | 9920 | 65 |
| Shanghai YuanYe Biotechnology Co., Ltd. | 15026964105 | 2881489226@qq.com | China | 89667 | 60 |
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| TargetMol Chemicals Inc. | +1-781-999-5354; +1-00000000000 | marketing@targetmol.com | United States | 32431 | 58 |
| InvivoChem | +1-708-310-1919 +1-13798911105 | sales@invivochem.cn | United States | 6378 | 58 |
| Shanghai Dongyang Biotechnology Co., Ltd. | 0512-13601744364 13601744364 | chemsharker@126.com | China | 1159 | 58 |
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