ChemicalBook >> CAS DataBase List >>N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methylthieno[2,3-d]pyrimidin-4-amine

N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methylthieno[2,3-d]pyrimidin-4-amine

CAS No.
452087-38-6
Chemical Name:
N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methylthieno[2,3-d]pyrimidin-4-amine
Synonyms
CIA1;CIA-1(Free base);CIA-1 (Free base);NR2F2-IN-1 free base;18:0 mPEG2000 PE sodium;N-(3,4-dimethoxyphenethyl)-6-methylthieno[2,3-d]pyrimidin-4-amine;N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methylthieno[2,3-d]pyrimidin-4-amine;Thieno[2,3-d]pyrimidin-4-amine, N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methyl-
CBNumber:
CB34625112
Molecular Formula:
C17H19N3O2S
Molecular Weight:
329.42
MDL Number:
MOL File:
452087-38-6.mol
MSDS File:
SDS
TDS File:
TDS
Last updated:2026-07-14 16:49:18

N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methylthieno[2,3-d]pyrimidin-4-amine Properties

Boiling point 529.6±50.0 °C(Predicted)
Density 1.264±0.06 g/cm3(Predicted)
pka 5.40±0.40(Predicted)
form Solid
color Light yellow to yellow

N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methylthieno[2,3-d]pyrimidin-4-amine price

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
ChemScene CS-1009304 NR2F2-IN-1 free base 99.34% 452087-38-6 5mg $162 2026-06-04 Buy
ChemScene CS-1009304 NR2F2-IN-1 free base 99.34% 452087-38-6 10mg $260 2026-06-04 Buy
ChemScene CS-1009304 NR2F2-IN-1 free base 99.34% 452087-38-6 25mg $520 2026-06-04 Buy
ChemScene CS-1009304 NR2F2-IN-1 free base 99.34% 452087-38-6 50mg $812 2026-06-04 Buy
ChemScene CS-1009304 NR2F2-IN-1 free base 99.34% 452087-38-6 100mg $1246 2026-06-04 Buy
Product number Packaging Price Buy
CS-1009304 5mg $162 Buy
CS-1009304 10mg $260 Buy
CS-1009304 25mg $520 Buy
CS-1009304 50mg $812 Buy
CS-1009304 100mg $1246 Buy

N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methylthieno[2,3-d]pyrimidin-4-amine Chemical Properties, Uses, Production

Uses

NR2F2-IN-1 (free base) is a potent and selective orphan nuclear receptor COUP-TFII (NR2F2) inhibitor. NR2F2-IN-1 (free base) substantially inhibits COUP-TFII–driven NGFIA reporter expression. NR2F2-IN-1 (free base) directly binds to the COUP-TFII ligand-binding domain and disrupts COUP-TFII interaction with transcription regulators, including FOXA1, thus repressing COUP-TFII activity on target gene regulation[1].

References

[1] Leiming Wang, et al. Small-molecule inhibitor targeting orphan nuclear receptor COUP-TFII for prostate cancer treatment. Sci Adv. 2020 Apr 29;6(18):eaaz8031. DOI:10.1126/sciadv.aaz8031

N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methylthieno[2,3-d]pyrimidin-4-amine Preparation Products And Raw materials

Raw materials

Preparation Products

N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methylthieno[2,3-d]pyrimidin-4-amine Suppliers

Global Suppliers ( 13)
Supplier Tel Email Country ProdList Advantage
Shanghai EFE Biological Technology Co., Ltd. 021-65675885 18964387627 info@efebio.com China 9799 58
Shanghai Yunpun industrial Co.,Ltd 21-61726900 15202122459; sales@yunpun.com China 497 58
TargetMol Chemicals Inc. +1-781-999-5354; +1-00000000000 marketing@targetmol.com United States 32431 58
Nantong QuanYi Biotechnology Co., Ltd 0513-66337626 18051384581 sales@chemhifuture.com China 5985 58
TargetMol Chemicals Inc. 15002134094 marketing@targetmol.cn China 29874 58
Aikon International Limited 025-58851090 19370895928 2850281427@qq.com China 8014 58
Shanghai Amole Biotechnology Co., Ltd. 13370042665 18916960931 2596183085@qq.com China 17234 58
ChemShuttle, Inc. 83588313 18800520310 sales@chemshuttle.com China 4999 58
Guangzhou Ruidi Biotechnology Co., Ltd. 020-82099279 18988941402 sales@ubiochem.com China 9998 58

View Latest Price from N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methylthieno[2,3-d]pyrimidin-4-amine manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
CIA-1 Free base pictures 2026-08-14 CIA-1 Free base
452087-38-6
$31.00-118.00 99.00% 10g TargetMol Chemicals Inc.
N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methylthieno[2,3-d]pyrimidin-4-amine CIA1 Thieno[2,3-d]pyrimidin-4-amine, N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methyl- CIA-1 (Free base) CIA-1(Free base) N-(3,4-dimethoxyphenethyl)-6-methylthieno[2,3-d]pyrimidin-4-amine 18:0 mPEG2000 PE sodium NR2F2-IN-1 free base 452087-38-6