GR 89696 FUMARATE
- CAS No.
- 126766-32-3
- Chemical Name:
- GR 89696 FUMARATE
- Synonyms
- GR 89696;GR 89696 FUMARATE;GR 89696 fumarate salt solid;GR 89696 fumarate, 10 mM in DMSO;Methyl 4-(2-(3,4-dichlorophenyl)acetyl)-3-(pyrrolidin-1-ylmethyl)piperazine-1-carboxylate fumarate;4-((3,4-Dichlorophenyl)acetyl)-3-(1-pyrrolidinylmethyl)-1-piperazinecarboxylicacidmethylesterfumarate;4-([3,4-DICHLOROPHENYL]ACETYL)-3-(1-PYRROLIDINYLMETHYL)-1-PIPERAZINECARBOXYLIC ACID METHYL ESTER FUMARATE
- CBNumber:
- CB4178514
- Molecular Formula:
- C23H29Cl2N3O7
- Molecular Weight:
- 530.4
- MDL Number:
- MFCD00274044
- MOL File:
- 126766-32-3.mol
- MSDS File:
- SDS
- TDS File:
- TDS
| storage temp. | Store at RT |
|---|---|
| solubility | ethanol: 4.0 mg/mL |
| form | solid |
| color | off-white |
| InChIKey | ABTNETSDXZBJTE-WLHGVMLRSA-N |
| SMILES | OC(=O)\C=C\C(O)=O.COC(=O)N1CCN(C(CN2CCCC2)C1)C(=O)Cc3ccc(Cl)c(Cl)c3 |
| FDA UNII | YDF52K5SDR |
| UNSPSC Code | 12352200 |
| NACRES | NA.77 |
SAFETY
Risk and Safety Statements
| PPE | Eyeshields, Gloves, type N95 (US) |
|---|---|
| WGK Germany | 3 |
| Storage Class | 11 - Combustible Solids |
GR 89696 FUMARATE price More Price(39)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Sigma-Aldrich | G133 | GR 89696 fumarate salt solid | 126766-32-3 | 25mg | $526 | 2026-04-30 | Buy |
| Cayman Chemical | 40145 | GR89696 (fumarate) ≥98% | 126766-32-3 | 5mg | $94 | 2026-04-30 | Buy |
| Cayman Chemical | 40145 | GR89696 (fumarate) ≥98% | 126766-32-3 | 10mg | $179 | 2026-04-30 | Buy |
| Cayman Chemical | 40145 | GR89696 (fumarate) ≥98% | 126766-32-3 | 25mg | $422 | 2026-04-30 | Buy |
| Cayman Chemical | 40145 | GR89696 (fumarate) ≥98% | 126766-32-3 | 50mg | $748 | 2026-04-30 | Buy |
GR 89696 FUMARATE Chemical Properties, Uses, Production
Uses
GR 89696 is a selective κ-opioid receptor agonist with anti-nociceptive and neuroprotective properties.
Biological Activity
Highly potent and selective κ -opioid agonist (IC 50 = 0.04 nM) that may be selective for the putative κ 2 receptor. Anti-nociceptive and neuroprotective in vivo .
in vivo
GR 89696 (intramuscular injection, 0.01-0.1 μg/kg) attenuates the scratching response induced by intrathecal morphine (0.03mg) in a dose-dependent manner without affecting the analgesic effect of morphine[1].
GR-896960(subcutaneous injection, 1 mg/kg) reduces cerebral artery infarct volume by 38% in a rat model of permanent focal ischemia[2].
storage
Store at +4°C
GR 89696 FUMARATE Preparation Products And Raw materials
Raw materials
Preparation Products
GR 89696 FUMARATE Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| 3B Pharmachem (Wuhan) International Co.,Ltd. | 18930552037 | 3bsc@sina.com | China | 15813 | 69 |
| BOC Sciences | 1-631-485-4226; 16314854226 | info@bocsci.com | United States | 9920 | 65 |
| Shanghai Lollane Biological Technology Co.,Ltd. | 021-52996696，15000506266 15000506266 | China | 4859 | 55 | |
| EMMX Biotechnology LLC | 888-539-0666 | info@emmx.com | United States | 8435 | 60 |
| Shanghai EFE Biological Technology Co., Ltd. | 021-65675885 18964387627 | info@efebio.com | China | 9799 | 58 |
| Shanghai YuanYe Biotechnology Co., Ltd. | 15026964105 | 2881489226@qq.com | China | 89667 | 60 |
| Shanghai Chaolan Chemical Technology Center | QQ：65489617 13301690235 | Sales@ATKchemical.com | China | 9699 | 58 |
| Shanghai Han-Xiang Chemical Co., Ltd. | 17754423994 | candy@biochempartner.com | China | 3057 | 58 |
| TargetMol Chemicals Inc. | +1-781-999-5354; +1-00000000000 | marketing@targetmol.com | United States | 32431 | 58 |
| Henan Weituxi Chemical Technology Co., Ltd. | 0371-63284658 18135795563 | 3905209149@qq.com | China | 9709 | 58 |
View Latest Price from GR 89696 FUMARATE manufacturers
| Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
|---|---|---|---|---|---|---|---|---|
 |
2026-07-15 | GR 89696 fumarate
126766-32-3
|
$58.00-155.00 | 99.84% | 10g | TargetMol Chemicals Inc. |
-
- GR 89696 fumarate
126766-32-3
- $58.00-155.00
- 99.84%
- TargetMol Chemicals Inc.
