Ramipril Diketopiperazine

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Ramipril Diketopiperazine Basic information
Product Name:Ramipril Diketopiperazine
Synonyms:[3S-[2(R*),3a,5ab,8ab,9ab]]-Decahydro-3-methyl-1,4-dioxo-a-(2-phenylethyl)-2H-cyclopenta[4,5]pyrrolo[1,2-a]pyrazine-2-acetic Acid Ethyl Ester;[3S-[2(R*),3a,5a,8a,9a]]-Decahydro-3-methyl-1,4-dioxo-a-(2-phenylethyl)-2H-cyclopenta[4,5]pyrrolo[1,2-a]pyrazine-2-acetic Acid Ethyl Ester;(αS,3S,5aS,8aS,9aS)-Decahydro-3-Methyl-1,4-dioxo-α-(2-phenylethyl)-2H-cyclopenta[4,5]pyrrolo[1,2-a]pyrazine-2-acetic Acid Ethyl Ester;[3S-[2(R*),3α,5aβ,8aβ,9aβ]]-Decahydro-3-Methyl-1,4-dioxo-α-(2-phenylethyl)-2H-cyclopenta[4,5]pyrrolo[1,2-a]pyrazine-2-acetic Acid Ethyl Ester;RaMipril IMpurity-D (EP);Ethyl (2S)2-[(3S,5aS,8aS, 9aS)-3-methyl-1,4-dioxodecahydro-1H-cyclopenta[e]pyrrolo[1,2-a]pyrazin-2-yl]-4-phenylbutanoate;Ethyl (2S)-2-[(3S,5aS,8aS,9aS)-3-methyl-1,4-dioxodecahydro-2H-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-2-yl]-4-phenyl butanoate;Ramipril Impurity 4(Ramipril EP Impurity D)
CAS:108731-95-9
MF:C23H30N2O4
MW:398.5
EINECS:
Product Categories:Aromatics;Chiral Reagents;Heterocycles;Intermediates & Fine Chemicals;Metabolites & Impurities;Pharmaceuticals
Mol File:108731-95-9.mol
Ramipril Diketopiperazine Structure
Ramipril Diketopiperazine Chemical Properties
Boiling point 597.4±50.0 °C(Predicted)
density 1.22±0.1 g/cm3(Predicted)
storage temp. 2-8°C
solubility DMSO: soluble,Ethanol: soluble
pka-1.16±0.40(Predicted)
Stability:Hygroscopic
Major Applicationpharmaceutical
InChIKeyKOVMAAYRBJCASY-JBDAPHQKSA-N
SMILESN21[C@@H]3[C@H](C[C@H]2C(=O)N([C@H](C1=O)C)[C@@H](CCc4ccccc4)C(=O)OCC)CCC3
Safety Information
WGK Germany WGK 3
Storage Class11 - Combustible Solids
MSDS Information
Ramipril Diketopiperazine Usage And Synthesis
UsesA metabolite of Ramipril (R111000).
UsesRamipril Diketopiperazine (Ramipril EP Impurity D) is a metabolite of Ramipril (R111000).
Ramipril Diketopiperazine Preparation Products And Raw materials
Tag:Ramipril Diketopiperazine(108731-95-9) Related Product Information
RAMIPRIL RELATED COMPOUND B (20 MG) (RAMIPRIL ISOPROPYLESTER) Ramipril Related Compound A (30 mg) ((2S,3aS,6aS)-1-[(S)2-[[(S)-1-(methoxycarbonyl)-3-phenylpropyl]amino]-1-oxopropyl]-octahydrocyclopenta[b]pyrrole-2-carboxylic acid) Ramiprilat (2R,3aR,6aR)- Ramipril Impurity 3 ((S,R,R)-2-Azabicyclo[3.3.0]octane-3 N-[(S)-(+)-1-(Ethoxycarbonyl)-3-phenylpropyl]-L-alanine Ramipril Impurity 1 ((R,S,S)-2-Azabicyclo[3.3.0]octane-3 Dibenzoyl-L-tartaric acid Ramiprilat Diketopiperazine Ramipril 1-Cyclopentyl-piperazin-2-one 5-(DIISOPROPYLAMINO)AMYLAMINE 1-Piperazineaceticacid,2-oxo-,methylester(8CI) H-Leu-Gly-OEt HCl (3-Oxo-1-piperazinyl)acetic acid Cyclo(-Leu-Gly) 3-Isobutyl-6-methyl-2,5-piperazinedione Ramipril Diketopiperazine