2(1H)-Pyridinone, 5-(3,5-dimethyl-4-isoxazolyl)-1-(phenylmethyl)-

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2(1H)-Pyridinone, 5-(3,5-dimethyl-4-isoxazolyl)-1-(phenylmethyl)- manufacturers

  • ZEN-2759
  • ZEN-2759 pictures
  • $39.00
  • 2026-06-09
  • CAS:1616400-50-0
  • Purity: 99.43%
  • Supply Ability: 10g
2(1H)-Pyridinone, 5-(3,5-dimethyl-4-isoxazolyl)-1-(phenylmethyl)- Basic information
Product Name:2(1H)-Pyridinone, 5-(3,5-dimethyl-4-isoxazolyl)-1-(phenylmethyl)-
Synonyms:2(1H)-Pyridinone, 5-(3,5-dimethyl-4-isoxazolyl)-1-(phenylmethyl)-;ZEN-2759;1-Benzyl-5-(3,5-dimethylisoxazol-4-yl)pyridin-2(1H)-one
CAS:1616400-50-0
MF:C17 H16 N2 O2
MW:280.32
EINECS:
Product Categories:
Mol File:1616400-50-0.mol
2(1H)-Pyridinone, 5-(3,5-dimethyl-4-isoxazolyl)-1-(phenylmethyl)- Structure
2(1H)-Pyridinone, 5-(3,5-dimethyl-4-isoxazolyl)-1-(phenylmethyl)- Chemical Properties
form Solid
color Off-white to light yellow
Safety Information
MSDS Information
2(1H)-Pyridinone, 5-(3,5-dimethyl-4-isoxazolyl)-1-(phenylmethyl)- Usage And Synthesis
DescriptionZEN-2759 is BRD4(BD1) inhibitor.
UsesZEN-2759 is a potent BET (Bromodomain and Extra-Terminal Domain) inhibitor, with IC50 values of 0.23, 0.08 and 0.28 μM for BRD4(BD1), BRD4(BD2), and BRD4(BD1BD2), respectively[1].
IC 50BRD4 (BD2): 0.08 μM (IC50); BRD4 (BD1): 0.23 μM (IC50); BRD4(BD1BD2): 0.28 μM (IC50)
References[1] Kharenko OA, et al. Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain (BET) Inhibitors Targeting a Methionine. J Med Chem. 2018 Sep 27;61(18):8202-8211. DOI:10.1021/acs.jmedchem.8b00666
2(1H)-Pyridinone, 5-(3,5-dimethyl-4-isoxazolyl)-1-(phenylmethyl)- Preparation Products And Raw materials
Tag:2(1H)-Pyridinone, 5-(3,5-dimethyl-4-isoxazolyl)-1-(phenylmethyl)-(1616400-50-0) Related Product Information
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