- OPIORPHIN
-
- $1.00
-
2026-10-12
- CAS:864084-88-8
- Min. Order: 1g
- Purity: 99%
- Supply Ability: 100kg
- OPIORPHIN
-
- $8.00
-
2026-09-02
- CAS:864084-88-8
- Min. Order: 1KG
- Purity: 99%
|
| | OPIORPHIN Basic information |
| Product Name: | OPIORPHIN | | Synonyms: | OPIORPHIN;H-Gln-Arg-Phe-Ser-Arg-OH;L-Arginine,L-glutaminyl-L-arginyl-L-phenylalanyl-L-seryl-;L-Glutaminyl-L-arginyl-L-phenylalanyl-L-seryl-L-arginine;opiorphin H-6504;L-glutamic acidaminoamideyl-L-argineaminoacyl-L-benzenepropylaminoacyl-L-serineaminoacyl-L-argineaminoacid;Opiorphin trifluoroacetate | | CAS: | 864084-88-8 | | MF: | C29H48N12O8 | | MW: | 692.77 | | EINECS: | | | Product Categories: | | | Mol File: | 864084-88-8.mol |  |
| | OPIORPHIN Chemical Properties |
| density | 1.51±0.1 g/cm3(Predicted) | | storage temp. | -20°C | | solubility | Methanol (Slightly), Water (Slightly) | | form | Solid | | pka | 3.23±0.10(Predicted) | | color | White to Off-White |
| | OPIORPHIN Usage And Synthesis |
| Uses | Opiorphin degrades enkephalin by inhibiting neutral endopeptidase and aminopeptidase N. Induces anorexic effect. | | Definition | ChEBI: Opiorphin is an oligopeptide. | | in vivo | Opiorphin (1.25-10 μg/kg; ICV; 0-60 min; male Kunming mice) induces potent analgesic effect in a dose- and time-dependent manner (ED50=3.22 μg/kg)[1]. | Animal Model: | Male Kunming mice[1] | | Dosage: | 1.25, 2.5, 5, 10 μg/kg | | Administration: | Intracerebroventrical injection; post-drug latency measurements were performed at 5, 10, 20, 30, 40, 50 and 60 min | | Result: | Had the percentage change of tail withdrawal latency (TWL) at 10 min after i.c.v. administration of 1.25-10 mg/kg was 28.90%, 44.37%, 56.43% and 91.899.79%, respectively. |
|
| | OPIORPHIN Preparation Products And Raw materials |
|