L-5,5-Dimethylthiazolidine-4-carboxylic acid

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L-5,5-Dimethylthiazolidine-4-carboxylic acid Basic information
Product Name:L-5,5-Dimethylthiazolidine-4-carboxylic acid
Synonyms:L-5,5-DIMETHYLTHIAZOLIDINE-4-CARBOXYLIC ACID;(R)-5,5-DIMETHYL-1,3-THIAZOLIDINE-4-CARBOXYLIC ACID;(R)-DTC-OH;(R)-5,5-Dimethyl-4-thiazolidinecarboxylic Acid;L-5,5-Dimethylthiazolidine-4-carboxyl;(R)-4-Carboxy-5,5-dimethylthiazolidine;(R)-5,5-Dimethylthiazolidine-4-carboxylic acid;(4R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid
CAS:72778-00-8
MF:C6H11NO2S
MW:161.22
EINECS:
Product Categories:All Inhibitors;Heterocycles;Inhibitors;Intermediates & Fine Chemicals;Pharmaceuticals;A - H;Amino Acids;Modified Amino Acids
Mol File:72778-00-8.mol
L-5,5-Dimethylthiazolidine-4-carboxylic acid Structure
L-5,5-Dimethylthiazolidine-4-carboxylic acid Chemical Properties
Melting point 206°C dec.
Boiling point 317.3±37.0 °C(Predicted)
density 1.195±0.06 g/cm3(Predicted)
refractive index [a]20D = - 149 ± 2 o (C=1 in water)
storage temp. 2-8°C
solubility Dichloromethane, DMSO, Methanol
form Solid
pka2.11±0.40(Predicted)
color White to off-white powder
InChIInChI=1S/C6H11NO2S/c1-6(2)4(5(8)9)7-3-10-6/h4,7H,3H2,1-2H3,(H,8,9)/t4-/m1/s1
InChIKeyPMQQFSDIECYOQV-SCSAIBSYSA-N
SMILESS1C(C)(C)[C@@H](C(O)=O)NC1
Safety Information
Hazard Codes Xi
Risk Statements 36/37/38
Safety Statements 26-36
WGK Germany 3
MSDS Information
ProviderLanguage
SigmaAldrich English
L-5,5-Dimethylthiazolidine-4-carboxylic acid Usage And Synthesis
Chemical PropertiesWhite Solid
UsesFound to act on the cell membrane of tumour cells, possible causing a reverse transformation to normal cells through restoration of contact inhibition.
Biological ActivityL-5,5-Dimethylthiazolidine-4-carboxylic acid (DTC) is used as a proline analog with restricted conformation in studies on receptor bound conformational requirements for agonists and antagonists of angiotensin II (ANG II).
L-5,5-Dimethylthiazolidine-4-carboxylic acid Preparation Products And Raw materials
Tag:L-5,5-Dimethylthiazolidine-4-carboxylic acid(72778-00-8) Related Product Information
Thiazolidine-4-carboxylic acid benzylpenicilloic acid L-2,2-DIMETHYLTHIAZOLIDINE-4-CARBOXYLIC ACID HYDROCHLORIDE 2-isopropyl-5,5-dimethylthiazolidine-4-carboxylic acid 5,5-dimethylthiazolidine-4-carboxylic acid (R)-3-(tert-Butoxycarbonyl)-2,2-dimethylthiazolidine-4-carboxylic acid Boc-(R)-5,5-dimethylthiazolidine-4-carboxylic acid penilloic acid 2-isopropyl-5,5-dimethylthiazolidine-4-carboxylic acid hydrochloride (R)-2,2-Dimethyl 4-thiazolidinecarboxylic acid hydrochloride L-5,5-Dimethylthiazolidine-4-carboxylic acid Fmoc-(R)-5,5-dimethylthiazolidine-4-carboxylic acid D-5,5-Dimethylthiazolidine-4-carboxylic acid) Bicyclo-[6, 5]-Boc-(2S, 3R)-Glu-(2S)-pen (4R)-3-tert-Butoxycarbonyl-2,2-dimethylthiazolidine-4-carboxylic acid Tobicillin (4S)-5,5-Dimethylthiazolidine-4-carboxylic acid Bicyclo-[6, 5]-Fmoc-(2S, 3R)-Glu-(2S)-pen