brepocitinib
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- $90 - $4766.8
- Product name: brepocitinib
- CAS: 1883299-62-4
- MF: C18H21F2N7O
- MW: 389.4
- EINECS:
- MDL Number:MFCD31813694
- Synonyms:PF-06700841 tosylate;((S)-2,2-difluorocyclopropyl)(3-(2-((1-methyl-1H-pyrazol-4-yl)amino)pyrimidin-4-yl)-3,8-diazabicyclo[3.2.1]octan-8-yl)methanone;PF 6700841;PF-06700841; PF 06700841; PF06700841; PF-6700841; PF 6700841; PF6700841; PF-06700841 TOSYLATE SALT;PF6700841;PF-6700841;CS-2861;Methanone, [(1S)-2,2-difluorocyclopropyl][3-[2-[(1-methyl-1H-pyrazol-4-yl)amino]-4-pyrimidinyl]-3,8-diazabicyclo[3.2.1]oct-8-yl]-
19 prices
Selected condition：
Brand
- ACHEMBLOCK
- Biorbyt Ltd
- Crysdot
- DC Chemicals
- Sigma-Aldrich
Package
- 5MG
- 25MG
- 100MG
- 250mg
- 1G
- ManufacturerACHEMBLOCK
- Product numberX189932
- Product descriptionPF-06700841 97.00%
- Packaging25MG
- Price$220
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberX189932
- Product descriptionPF-06700841 97.00%
- Packaging25MG
- Price$220
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberX189932
- Product descriptionPF-06700841 97.00%
- Packaging5MG
- Price$90
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberX189932
- Product descriptionPF-06700841 97.00%
- Packaging5MG
- Price$90
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberX189932
- Product descriptionPF-06700841 97.00%
- Packaging100MG
- Price$570
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberX189932
- Product descriptionPF-06700841 97.00%
- Packaging100MG
- Price$570
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberX189932
- Product descriptionPF-06700841 97.00%
- Packaging1G
- Price$1940
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberX189932
- Product descriptionPF-06700841 97.00%
- Packaging1G
- Price$1940
- Updated2026-05-27
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb573132
- Product descriptionPF-06700841 tosylate >98%
- Packaging250mg
- Price$2245.7
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb573132
- Product descriptionPF-06700841 tosylate >98%
- Packaging100mg
- Price$1283.5
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb573132
- Product descriptionPF-06700841 tosylate >98%
- Packaging1g
- Price$4766.8
- Updated2021-12-16
- Buy
- ManufacturerCrysdot
- Product numberCD31005024
- Product description4-[(1R,5S)-8-[(1S)-2,2-difluorocyclopropanecarbonyl]-3,8-diazabicyclo[3.2.1]octan-3-yl]-N-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine 98%
- Packaging25mg
- Price$480
- Updated2021-12-16
- Buy
- ManufacturerCrysdot
- Product numberCD31005024
- Product description4-[(1R,5S)-8-[(1S)-2,2-difluorocyclopropanecarbonyl]-3,8-diazabicyclo[3.2.1]octan-3-yl]-N-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine 98%
- Packaging25mg
- Price$480
- Updated2026-05-27
- Buy
- ManufacturerDC Chemicals
- Product numberDC12489
- Product descriptionPF-06700841 free base >98%
- Packaging100mg
- Price$850
- Updated2026-05-24
- Buy
- ManufacturerDC Chemicals
- Product numberDC12489
- Product descriptionPF-06700841freebase >98%
- Packaging250mg
- Price$1500
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC12489
- Product descriptionPF-06700841 free base >98%
- Packaging250mg
- Price$1500
- Updated2026-05-24
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| ACHEMBLOCK | X189932 | PF-06700841 97.00% | 25MG | $220 | 2026-05-25 | Buy |
| ACHEMBLOCK | X189932 | PF-06700841 97.00% | 25MG | $220 | 2026-05-27 | Buy |
| ACHEMBLOCK | X189932 | PF-06700841 97.00% | 5MG | $90 | 2026-05-25 | Buy |
| ACHEMBLOCK | X189932 | PF-06700841 97.00% | 5MG | $90 | 2026-05-27 | Buy |
| ACHEMBLOCK | X189932 | PF-06700841 97.00% | 100MG | $570 | 2026-05-25 | Buy |
| ACHEMBLOCK | X189932 | PF-06700841 97.00% | 100MG | $570 | 2026-05-27 | Buy |
| ACHEMBLOCK | X189932 | PF-06700841 97.00% | 1G | $1940 | 2026-05-25 | Buy |
| ACHEMBLOCK | X189932 | PF-06700841 97.00% | 1G | $1940 | 2026-05-27 | Buy |
| Biorbyt Ltd | orb573132 | PF-06700841 tosylate >98% | 250mg | $2245.7 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb573132 | PF-06700841 tosylate >98% | 100mg | $1283.5 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb573132 | PF-06700841 tosylate >98% | 1g | $4766.8 | 2021-12-16 | Buy |
| Crysdot | CD31005024 | 4-[(1R,5S)-8-[(1S)-2,2-difluorocyclopropanecarbonyl]-3,8-diazabicyclo[3.2.1]octan-3-yl]-N-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine 98% | 25mg | $480 | 2021-12-16 | Buy |
| Crysdot | CD31005024 | 4-[(1R,5S)-8-[(1S)-2,2-difluorocyclopropanecarbonyl]-3,8-diazabicyclo[3.2.1]octan-3-yl]-N-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine 98% | 25mg | $480 | 2026-05-27 | Buy |
| DC Chemicals | DC12489 | PF-06700841 free base >98% | 100mg | $850 | 2026-05-24 | Buy |
| DC Chemicals | DC12489 | PF-06700841freebase >98% | 250mg | $1500 | 2021-12-16 | Buy |
| DC Chemicals | DC12489 | PF-06700841 free base >98% | 250mg | $1500 | 2026-05-24 | Buy |
Properties
Boiling point :637.1±65.0 °C(Predicted)
Density :1.63±0.1 g/cm3(Predicted)
storage temp. :room temp
solubility :DMSO: 78 mg/mL (200.31 mM);Ethanol: 78 mg/mL (200.31 mM)
form :powder
pka :7.28±0.10(Predicted)
color :white to beige
Water Solubility :Water: Insoluble
InChIKey :BUWBRTXGQRBBHG-RUXDESIVSA-N
SMILES :C([C@@H]1CC1(F)F)(N1C2CCC1CN(C1C=CN=C(NC3=CN(C)N=C3)N=1)C2)=O
Density :1.63±0.1 g/cm3(Predicted)
storage temp. :room temp
solubility :DMSO: 78 mg/mL (200.31 mM);Ethanol: 78 mg/mL (200.31 mM)
form :powder
pka :7.28±0.10(Predicted)
color :white to beige
Water Solubility :Water: Insoluble
InChIKey :BUWBRTXGQRBBHG-RUXDESIVSA-N
SMILES :C([C@@H]1CC1(F)F)(N1C2CCC1CN(C1C=CN=C(NC3=CN(C)N=C3)N=1)C2)=O
Safety Information
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Description
PF-06700841 tosylate salt has been used as an inhibitor of Janus kinase1 (JAK1) to study its therapeutic effect on the adjuvant induced arthritis (AIA) rat model. It has also been used as an inhibitor of interferon-α/β receptor alpha chain (IFNAR1) signaling adaptor tyrosine kinase (2TYK2) in mice.More related product prices
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