ChemicalBook >> CAS DataBase List >>AP-761

AP-761

CAS No.
1093108-50-9
Chemical Name:
AP-761
Synonyms
AP-761;BI671800;BI-67180;BI-671800 ,S0495;AP-761 / BI671800;BI-671800 (Actimis);BI 671800 (BI671800);BI-671800, 10 mM in DMSO;BI671800;AP-761;AP761;AP 761;BI-671800,BI671800,Inhibitor,BI 671800,Prostaglandin Receptor,inhibit
CBNumber:
CB32728622
Molecular Formula:
C25H26F3N5O3
Molecular Weight:
501.5
MDL Number:
MOL File:
1093108-50-9.mol
MSDS File:
SDS
Last updated:2026-04-16 17:44:27
Product description Number Pack Size Price
BI-671800 27638 5mg $692
BI-671800 27638 10mg $1169
BI-671800 27638 1mg $214
BI-671800 B591753 2.5mg $565
BI-671800 99.06% CS-0070031 100mg $2650

AP-761 Properties

Boiling point 611.4±55.0 °C(Predicted)
Density 1.351±0.06 g/cm3(Predicted)
storage temp. 4°C, protect from light
solubility DMSO: soluble
form A crystalline solid
pka 3.20±0.10(Predicted)
color White to off-white
FDA UNII 721F767LHB

AP-761 price More Price(14)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Cayman Chemical 27638 BI-671800 1093108-50-9 5mg $692 2024-03-01 Buy
Cayman Chemical 27638 BI-671800 1093108-50-9 10mg $1169 2024-03-01 Buy
Cayman Chemical 27638 BI-671800 1093108-50-9 1mg $214 2024-03-01 Buy
TRC B591753 BI-671800 1093108-50-9 2.5mg $565 2021-12-16 Buy
ChemScene CS-0070031 BI-671800 99.06% 1093108-50-9 100mg $2650 2021-12-16 Buy
Product number Packaging Price Buy
27638 5mg $692 Buy
27638 10mg $1169 Buy
27638 1mg $214 Buy
B591753 2.5mg $565 Buy
CS-0070031 100mg $2650 Buy

AP-761 Chemical Properties,Uses,Production

Uses

BI-671800 is a selective and potent CRTH2 antagonist.

in vivo

BI-671800 (compound A, 0.1-10 mg/kg, i.g.) shows significant inhibition of AHR in mice[1].
BI-671800 (compound A), effectively blocks edema formation and greatly reduces the inflammatory infiltrate and skin pathology observed in drug vehicle-treated animals[3].

Animal Model:6-8-week-old age- and sex-matched BALB/c mice (mice were sensitized for 14 days, challenged intranasally)[1].
Dosage:10-0.1 mg/kg
Administration:Oral gavage for 4 weeks
Result:Shows significant inhibition of AHR in mice.

IC 50

hCRTH2: 4.5 nM (IC50); mCRTH2: 3.7 μM (IC50)

AP-761 Preparation Products And Raw materials

Raw materials

Preparation Products

AP-761 Suppliers

Global( 55)Suppliers
Supplier Tel Email Country ProdList Advantage
career henan chemical co
+86-0371-86658258 +8613203830695 factory@coreychem.com China 29794 58
TargetMol Chemicals Inc.
+1-781-999-5354; +17819995354 marketing@targetmol.com United States 32467 58
Nantong HI-FUTURE Biology Co., Ltd.
+undefined18051384581 sales@chemhifuture.com China 3135 58
TargetMol Chemicals Inc.
+1-781-999-5354; support@targetmol.com United States 39040 58
Aladdin Scientific
tp@aladdinsci.com United States 57505 58
BOC Sciences 1-631-485-4226; 16314854226 info@bocsci.com United States 12952 65
Taizhou Tongxin Bio-Tech Co., Ltd 0523-86818997 18652728585 sales@allyrise.com China 2976 60
Bide Pharmatech Ltd. 400-400-164-7117 18317119277 product02@bidepharm.com China 40000 60
Shanghaizehan biopharma technology co., Ltd. 021-61350663 13052117465 sales@zehanbiopharma.com China 979 55
Taizhou Ruixin Chemical Co., Ltd. 0576-89085261 15867635987 jasonhu09@163.com China 442 50

View Lastest Price from AP-761 manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
BI-671800 pictures 2026-04-16 BI-671800
1093108-50-9
US $44.00-179.00 / mg 99.19% 10g TargetMol Chemicals Inc.
BI-671800 pictures 2026-04-16 BI-671800
1093108-50-9
US $44.00-179.00 / mg 99.19% 10g TargetMol Chemicals Inc.
AP-761 pictures 2020-01-09 AP-761
1093108-50-9
US $2.00 / KG 1g 98%min ask Career Henan Chemical Co
  • BI-671800 pictures
  • BI-671800
    1093108-50-9
  • US $44.00-179.00 / mg
  • 99.19%
  • TargetMol Chemicals Inc.
  • BI-671800 pictures
  • BI-671800
    1093108-50-9
  • US $44.00-179.00 / mg
  • 99.19%
  • TargetMol Chemicals Inc.
  • AP-761 pictures
  • AP-761
    1093108-50-9
  • US $2.00 / KG
  • 98%min
  • Career Henan Chemical Co

AP-761 Spectrum

AP-761 5-Pyrimidineacetic acid, 4,6-bis(dimethylamino)-2-[[4-[[4-(trifluoromethyl)benzoyl]amino]phenyl]methyl]- BI671800 BI671800;AP-761;AP761;AP 761 BI 671800 (BI671800) AP-761 / BI671800 BI-67180 BI-671800,BI671800,Inhibitor,BI 671800,Prostaglandin Receptor,inhibit BI-671800 (Actimis) 2-(4,6-Bis(dimethylamino)-2-(4-(4-(trifluoromethyl)benzamido)benzyl)pyrimidin-5-yl)acetic acid BI-671800, 10 mM in DMSO BI-671800 ,S0495 1093108-50-9 AP-761