ChemicalBook >> CAS DataBase List >>AP-761
AP-761
- CAS No.
- 1093108-50-9
- Chemical Name:
- AP-761
- Synonyms
- AP-761;BI671800;BI-67180;BI-671800 ,S0495;AP-761 / BI671800;BI-671800 (Actimis);BI 671800 (BI671800);BI-671800, 10 mM in DMSO;BI671800;AP-761;AP761;AP 761;BI-671800,BI671800,Inhibitor,BI 671800,Prostaglandin Receptor,inhibit
- CBNumber:
- CB32728622
- Molecular Formula:
- C25H26F3N5O3
- Molecular Weight:
- 501.5
- MDL Number:
- MOL File:
- 1093108-50-9.mol
- MSDS File:
- SDS
Last updated:2026-04-16 17:44:27
| Product description | Number | Pack Size | Price |
| BI-671800 | 27638 | 5mg | $692 |
| BI-671800 | 27638 | 10mg | $1169 |
| BI-671800 | 27638 | 1mg | $214 |
| BI-671800 | B591753 | 2.5mg | $565 |
| BI-671800 99.06% | CS-0070031 | 100mg | $2650 |
| Boiling point | 611.4±55.0 °C(Predicted) |
|---|---|
| Density | 1.351±0.06 g/cm3(Predicted) |
| storage temp. | 4°C, protect from light |
| solubility | DMSO: soluble |
| form | A crystalline solid |
| pka | 3.20±0.10(Predicted) |
| color | White to off-white |
| FDA UNII | 721F767LHB |
AP-761 price More Price(14)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Cayman Chemical | 27638 | BI-671800 | 1093108-50-9 | 5mg | $692 | 2024-03-01 | Buy |
| Cayman Chemical | 27638 | BI-671800 | 1093108-50-9 | 10mg | $1169 | 2024-03-01 | Buy |
| Cayman Chemical | 27638 | BI-671800 | 1093108-50-9 | 1mg | $214 | 2024-03-01 | Buy |
| TRC | B591753 | BI-671800 | 1093108-50-9 | 2.5mg | $565 | 2021-12-16 | Buy |
| ChemScene | CS-0070031 | BI-671800 99.06% | 1093108-50-9 | 100mg | $2650 | 2021-12-16 | Buy |
AP-761 Chemical Properties,Uses,Production
Uses
BI-671800 is a selective and potent CRTH2 antagonist.
in vivo
BI-671800 (compound A, 0.1-10 mg/kg, i.g.) shows significant inhibition of AHR in mice[1].
BI-671800 (compound A), effectively blocks edema formation and greatly reduces the inflammatory infiltrate and skin pathology observed in drug vehicle-treated animals[3].
| Animal Model: | 6-8-week-old age- and sex-matched BALB/c mice (mice were sensitized for 14 days, challenged intranasally)[1]. |
| Dosage: | 10-0.1 mg/kg |
| Administration: | Oral gavage for 4 weeks |
| Result: | Shows significant inhibition of AHR in mice. |
IC 50
hCRTH2: 4.5 nM (IC50); mCRTH2: 3.7 μM (IC50)
AP-761 Preparation Products And Raw materials
Raw materials
Preparation Products
AP-761 Suppliers
Global( 55)Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| career henan chemical co | +86-0371-86658258 +8613203830695 | factory@coreychem.com | China | 29794 | 58 |
| TargetMol Chemicals Inc. | +1-781-999-5354; +17819995354 | marketing@targetmol.com | United States | 32467 | 58 |
| Nantong HI-FUTURE Biology Co., Ltd. | +undefined18051384581 | sales@chemhifuture.com | China | 3135 | 58 |
| TargetMol Chemicals Inc. | +1-781-999-5354; | support@targetmol.com | United States | 39040 | 58 |
| Aladdin Scientific | tp@aladdinsci.com | United States | 57505 | 58 | |
| BOC Sciences | 1-631-485-4226; 16314854226 | info@bocsci.com | United States | 12952 | 65 |
| Taizhou Tongxin Bio-Tech Co., Ltd | 0523-86818997 18652728585 | sales@allyrise.com | China | 2976 | 60 |
| Bide Pharmatech Ltd. | 400-400-164-7117 18317119277 | product02@bidepharm.com | China | 40000 | 60 |
| Shanghaizehan biopharma technology co., Ltd. | 021-61350663 13052117465 | sales@zehanbiopharma.com | China | 979 | 55 |
| Taizhou Ruixin Chemical Co., Ltd. | 0576-89085261 15867635987 | jasonhu09@163.com | China | 442 | 50 |
View Lastest Price from AP-761 manufacturers
| Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
|---|---|---|---|---|---|---|---|---|
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2026-04-16 | BI-671800
1093108-50-9
|
US $44.00-179.00 / mg | 99.19% | 10g | TargetMol Chemicals Inc. | ||
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2026-04-16 | BI-671800
1093108-50-9
|
US $44.00-179.00 / mg | 99.19% | 10g | TargetMol Chemicals Inc. | ||
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2020-01-09 | AP-761
1093108-50-9
|
US $2.00 / KG | 1g | 98%min | ask | Career Henan Chemical Co |
1093108-50-9(AP-761)Related Search:
AP-761
5-Pyrimidineacetic acid, 4,6-bis(dimethylamino)-2-[[4-[[4-(trifluoromethyl)benzoyl]amino]phenyl]methyl]-
BI671800
BI671800;AP-761;AP761;AP 761
BI 671800
(BI671800)
AP-761 / BI671800
BI-67180
BI-671800,BI671800,Inhibitor,BI 671800,Prostaglandin Receptor,inhibit
BI-671800 (Actimis)
2-(4,6-Bis(dimethylamino)-2-(4-(4-(trifluoromethyl)benzamido)benzyl)pyrimidin-5-yl)acetic acid
BI-671800, 10 mM in DMSO
BI-671800 ,S0495
1093108-50-9
AP-761







