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4-Bromoindole-2-carboxylic acid methyl ester

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4-Bromoindole-2-carboxylic acid methyl ester Basic information
Product Name:4-Bromoindole-2-carboxylic acid methyl ester
Synonyms:1H-Indole-2-carboxylic acid, 4-broMo-, Methyl ester;4-bromo-1H-indole-2-carboxylic acid methyl ester;4-Bromoindole-2-carboxylic acid methyl ester;Methyl 4-bromoindole-2-carboxylate;Methyl 4-bromo-1H-indole-2-carboxylate 98%;methyl 4-bromo-1H-indole-2-carboxylate - [M83515]
CAS:167479-13-2
MF:C10H8BrNO2
MW:254.08
EINECS:
Product Categories:
Mol File:167479-13-2.mol
4-Bromoindole-2-carboxylic acid methyl ester Structure
4-Bromoindole-2-carboxylic acid methyl ester Chemical Properties
Boiling point 386.2±22.0 °C(Predicted)
density 1.629±0.06 g/cm3(Predicted)
storage temp. Sealed in dry,Room Temperature
pka14.04±0.30(Predicted)
form solid
color Beige
Safety Information
HazardClass IRRITANT
HS Code 2924297099
MSDS Information
4-Bromoindole-2-carboxylic acid methyl ester Usage And Synthesis
Synthesis
2-Propenoic acid, 2-azido-3-(2-bromophenyl)-, methyl ester

220448-44-2

4-Bromoindole-2-carboxylic acid methyl ester

167479-13-2

GENERAL METHOD: Methyl 3-aryl-2-azidoacrylate (20.0 mmol) was added in a single addition to a pre-heated to reflux xylene solution (75 mL) and the reaction was kept at reflux for 2 hours. Upon completion of the reaction, the solvent was removed by rotary evaporator. The resulting residue was purified by silica gel column chromatography with mixed petroleum ether/ethyl acetate solvent as eluent. The synthesis of compounds 12, 18 and 19 has been reported in the literature [9b, 13, 14].

References[1] European Journal of Medicinal Chemistry, 2012, vol. 49, p. 379 - 396
4-Bromoindole-2-carboxylic acid methyl ester Preparation Products And Raw materials
Raw materials2-Propenoic acid, 2-azido-3-(2-bromophenyl)-, methyl ester
Tag:4-Bromoindole-2-carboxylic acid methyl ester(167479-13-2) Related Product Information
4-Bromooxindole 4-Bromoindole-1-carboxylic acid tert-butyl ester 4-Bromoindole-2-carboxylic acid ethyl ester Ethyl4-(bromomethyl)-3-nitrobenzoate Indole methyl 4-bromo-1H-indole-3-carboxylate 1H-Indazole-3-carboxaldehyde, 4-broMo- 4-Bromoindole-3-carboxaldehyde 4-Bromo-2-indolecarboxylic acid 1H-Indole-3-aceticacid,4-bromo-(9CI) 4-Bromoindole 4-Bromoindole-2-carboxylic acid methyl ester 1H-Indole-2-carboxylic acid,4-bromo-3-formyl-,ethyl ester Ethyl 4-bromo-5-methoxy-1H-indole-2-carboxylate 5-Bromo-8H-1,3-dioxa-8-aza-as-indacene-7-carboxylic acid methyl ester 4-Bromo-7-ethoxy-6-methoxy-1H-indole-2-carboxylic acid methyl ester 4-Bromo-6,7-dimethoxy-1H-indole-2-carboxylic acid methyl ester