TFLLR-NH2

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Company Name: BOC Sciences
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Products Intro: Product Name:TFLLR-NH2
CAS:197794-83-5
Purity:98% Package:5 mg Remarks:Reach out to us for more information about custom solutions.
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Products Intro: Product Name:TFLLR-NH2
CAS: 197794-83-5
Purity:99% Package:1KG;7USD
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Products Intro: Product Name:TFLLR-NH2 2TFA(197794-83-5(free base))
CAS:197794-83-5
Purity:99.56% Package:1mg;133USD|5mg;515USD|10mg;743USD Remarks:REAGENT;FOR LABORATORY USE ONLY
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Products Intro: Product Name:TFLLR-NH2(2TFA)
CAS:197794-83-5
Purity:99% Package:10kg 25kg 200 kilograms per barrel Remarks:good
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Products Intro: CAS:197794-83-5
Purity:99% Package:5KG;1KG

TFLLR-NH2 manufacturers

  • TFLLR-NH2
  • TFLLR-NH2 pictures
  • $0.00 / 1kg
  • 2025-04-04
  • CAS:197794-83-5
  • Min. Order: 1kg
  • Purity: 98%
  • Supply Ability: 1Ton
  • TFLLR-NH2
  • TFLLR-NH2 pictures
  • $7.00 / 1KG
  • 2020-02-14
  • CAS: 197794-83-5
  • Min. Order: 1KG
  • Purity: 99%
  • Supply Ability: 100KG
TFLLR-NH2 Basic information
Product Name:TFLLR-NH2
Synonyms:H-THR-PHE-LEU-LEU-ARG-NH2;THR-PHE-LEU-LEU-ARG-NH2;THROMBIN RECEPTOR (PAR-1), HYBRIDE HUMAN-XENOPE;TFLLR-AMIDE;TFLLR-NH2;(Thr1)-TRAP-5 amide;TFLLR-NH2 Protease-Activated Receptor 1 (PAR1) Agonist;(2S)-N-[(2S)-1-[[(2S)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]-2-[[(2S)-2-[[(2S,3R)-2-amino-3-hydroxybutanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanamide
CAS:197794-83-5
MF:C31H53N9O6
MW:647.81
EINECS:
Product Categories:Proteinase-activated receptor (PAR);Peptide Receptors
Mol File:197794-83-5.mol
TFLLR-NH2 Structure
TFLLR-NH2 Chemical Properties
density 1.31±0.1 g/cm3(Predicted)
storage temp. Desiccate at -20°C
form Powder
pka12.10±0.45(Predicted)
Water Solubility Soluble to 1 mg/ml in water
SequenceThr-Phe-Leu-Leu-Arg-NH2
Safety Information
MSDS Information
TFLLR-NH2 Usage And Synthesis
UsesTFLLR-NH2 is a PAR-1 activator.
in vivo

Injection of TF-NH2 into the rat paw stimulates a marked and sustained oedema. An NK1R antagonist and ablation of sensory nerves with capsaicin inhibit oedema by 44% at 1h and completely by 5h. In wild-type but not PAR1/ mice, TF-NH2 stimulates Evans blue extravasation in the bladder, oesophagus, stomach, intestine and pancreas by 2–8 fold. Extravasation in the bladder, oesophagus and stomach is abolished by an NK1R antagonist[1]. TFp-NH2 produces notable contraction at 3-50 μM and relaxation at 0.3-50 μM, in the absence of apamin. The concentration-response curve for TFp-NH2-induced contraction is remarkably shifted left, when the TFp-NH2-induced relaxation is blocked by apamin at 0.1 μM[3].

IC 50PAR1: 1.9 μM (EC50)
storage-20°C
TFLLR-NH2 Preparation Products And Raw materials
Tag:TFLLR-NH2(197794-83-5) Related Product Information
DL-Threonine hydrate(2:1) ANTI HUMAN TR-ALPHA Trifluoroacetamide H-SER-PHE-LEU-LEU-ARG-NH2 TFLLR-NH2 H-THR-PHE-LEU-LEU-ARG-NH2 TRIFLUOROACETATE SALT THR-PHE-LEU-LEU-ARG-ASN-PRO-ASN-ASP-LYS-NH2