GABAA receptor agent 5 NEW
| Price | $1520 | $1980 | $2500 |
| Package | 25mg | 50mg | 100mg |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2025-10-27 |
Product Details
| Product Name: GABAA receptor agent 5 | CAS No.: 1808389-92-5 |
| Supply Ability: 10g | Release date: 2025/10/27 |
Product Introduction
Bioactivity
| Name | GABAA receptor agent 5 |
| Description | GABAA Receptor Agent 5 (compound 018) serves as a potent γ-GABAAR antagonist, possessing a Ki of 0.020 μM. This compound exhibits γ-GABAAR antagonist properties, yet it demonstrates low cellular membrane permeability [1]. |
| In vitro | Compound 018, a GABAA receptor agent, exhibits antagonist activity, demonstrated by its IC50 values. These are 0.24 μM for α1β2δ, 0.088 μM for α4β1δ, 0.068 μM for α4β2δ, 0.33 μM for α6β2δ, 0.79 μM for α1β2γ2, 0.32 μM for α2β2γ2, 0.079 μM for α3β2γ2, and 0.051 μM for α5β2γ2 subtypes, respectively [1]. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Inhibitors Related | Compound PDK0243 | p-Hydroxybenzaldehyde | Urethane | Baicalin | Penicillin G sodium salt | DL-Pyroglutamic acid | Valproic Acid | Halothane | Chlorothymol | (-)-α-Pinene | Dihydromyricetin | Methionine |
Company Profile Introduction
TargetMol Chemicals Inc. is headquartered in Boston, MA, and specializes in products and services that serve the research needs of chemical and biological scientists worldwide. With a client base in 40+ countries, TargetMol has evolved into one of the biggest global research suppliers for compound libraries and small molecule compounds.
170+ Compound Libraries， 10000+ Noval Small Molecucles，16000+ Nature Compounds
TargetMol diligently updates and offers over 170 types of compound libraries and a wide range of high-quality research chemicals, including inhibitors, activators, natural products, peptides, antibodies , and novel life-science kits for laboratory and scientific use. In addition, our lab allows us to conduct CADD (computer-aided drug design) and chemical synthesis to meet the customization needs of our clients.
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United States- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, Massachusetts, USA
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