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Epinastine hydrobromide

CAS No.
127786-29-2
Chemical Name:
Epinastine hydrobromide
Synonyms
EPINASTIN HBR;Epinastine HBr;Epinastine-13C-d3 HBr;Epinastin hydrobromide;epinastine hydrobromide;9,13b-Dihydro-1H-dibenzo[c,f]imidazo[1,5-a]azepin-3-amine hydrobromide;9,13b-dihydro-1H-dibenz[c,f]imidazo[1,5-a]azepin-3-amine monohydrobromide;(+/-)-3-amino-9,13b-dihydro-1h-dibenz[c,f]imidazo[1,5-a]azepine hydrobromide;6-Aminomethyl-6,11-dihydro-5H-dibenz[b,e]azepine (E)-2-butenedioate Epinastine hydrobromide
CBNumber:
CB2854847
Molecular Formula:
C16H16BrN3
Molecular Weight:
330.22234
MDL Number:
MOL File:
127786-29-2.mol
Last updated:2025-07-04 15:21:27
Product description Number Pack Size Price
EpinastinHbr E589593 50mg $75
EPINASTINE HYDROBROMIDE 95.00% API0025691 5MG $505.47
EPINASTINE HYDROBROMIDE 95.00% API0025691 1G $1274.7
9,13b-Dihydro-1H-dibenzo[c,f]imidazo[1,5-a]azepin-3-aminehydrobromide 127786292 1g $568
9,13b-Dihydro-1H-dibenzo[c,f]imidazo[1,5-a]azepin-3-aminehydrobromide 95+% CD31004008 1g $705
More product size

Epinastine hydrobromide Properties

Melting point 284-286°
storage temp. Sealed in dry,Room Temperature
InChI InChI=1S/C16H15N3.BrH/c17-16-18-10-15-13-7-3-1-5-11(13)9-12-6-2-4-8-14(12)19(15)16;/h1-8,15H,9-10H2,(H2,17,18);1H
InChIKey ADPMHRDERZTFIN-UHFFFAOYSA-N
SMILES N12C(N)=NCC1C1C=CC=CC=1CC1C=CC=CC2=1.Br
FDA UNII 4O6LIW7G3N

SAFETY

Risk and Safety Statements

Symbol(GHS)  GHS hazard pictograms
GHS07
Signal word  Warning
Hazard statements  H302
Precautionary statements  P264-P270-P301+P312-P330-P501

Epinastine hydrobromide price

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
TRC E589593 EpinastinHbr 127786-29-2 50mg $75 2021-12-16 Buy
American Custom Chemicals Corporation API0025691 EPINASTINE HYDROBROMIDE 95.00% 127786-29-2 5MG $505.47 2021-12-16 Buy
American Custom Chemicals Corporation API0025691 EPINASTINE HYDROBROMIDE 95.00% 127786-29-2 1G $1274.7 2021-12-16 Buy
Alichem 127786292 9,13b-Dihydro-1H-dibenzo[c,f]imidazo[1,5-a]azepin-3-aminehydrobromide 127786-29-2 1g $568 2021-12-16 Buy
Crysdot CD31004008 9,13b-Dihydro-1H-dibenzo[c,f]imidazo[1,5-a]azepin-3-aminehydrobromide 95+% 127786-29-2 1g $705 2021-12-16 Buy
Product number Packaging Price Buy
E589593 50mg $75 Buy
API0025691 5MG $505.47 Buy
API0025691 1G $1274.7 Buy
127786292 1g $568 Buy
CD31004008 1g $705 Buy

Epinastine hydrobromide Chemical Properties,Uses,Production

Application

Clinical studies have shown that, at the same dosage, epinastine hydrochloride is significantly more effective than other second-generation histamine H1 receptor antagonists such as terfenadine, astamiva, and ketotifen, and also has a lower incidence of central sedation and cardiotoxicity. Therefore, the market demand for epinastine hydrochloride is substantial, making its synthesis necessary. Literature searches reveal that publicly available patents and literature use 6-aminomethyl-6,11-dihydro-5H-dibenzo[b,e]azapyridine (Ⅳ) as a key intermediate in epinastine synthesis, which is cyclized with cyanogen bromide to yield epinastine. Epinastine hydrobromide is also a synthetic intermediate for epinastine.

Epinastine hydrobromide Preparation Products And Raw materials

Raw materials

Preparation Products

Global( 53)Suppliers
Supplier Tel Email Country ProdList Advantage
Henan Tianfu Chemical Co.,Ltd.
+86-0371-55170693 +86-19937530512 info@tianfuchem.com China 21599 55
Nanjing Dolon Biotechnology Co.,Ltd.
18905173768 52513593@qq.com CHINA 2972 58
BOC Sciences
+1-631-485-4226 inquiry@bocsci.com United States 19552 58
CONIER CHEM AND PHARMA LIMITED
+8618523575427 sales@conier.com China 49977 58
career henan chemical co
+86-0371-86658258 +8613203830695 factory@coreychem.com China 29795 58
AFINE CHEMICALS LIMITED
+86-0571-85134551 sales@afinechem.com China 15082 58
Dayang Chem (Hangzhou) Co.,Ltd.
+86-0571-88938639 +8617705817739 info@dycnchem.com China 52846 58
Hebei Chuanghai Biotechnology Co., Ltd
+8615531151365 mina@chuanghaibio.com China 18126 58
PT CHEM GROUP LIMITED
+86-85511178; peter68@ptchemgroup.com China 35425 58
GIHI CHEMICALS CO.,LIMITED
+86-571-86217390; +8618058761490 info@gihichemicals.com China 49958 58

View Lastest Price from Epinastine hydrobromide manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
Epinastine hydrobromide pictures 2020-01-08 Epinastine hydrobromide
127786-29-2
US $2.00 / KG 1KG 98% 100g , 1kg, 5kg , 50kg Career Henan Chemical Co
Epinastine-13C-d3 HBr (+/-)-3-amino-9,13b-dihydro-1h-dibenz[c,f]imidazo[1,5-a]azepine hydrobromide EPINASTIN HBR Epinastine HBr 9,13b-Dihydro-1H-dibenzo[c,f]imidazo[1,5-a]azepin-3-amine hydrobromide epinastine hydrobromide Epinastin hydrobromide 6-Aminomethyl-6,11-dihydro-5H-dibenz[b,e]azepine (E)-2-butenedioate Epinastine hydrobromide 9,13b-dihydro-1H-dibenz[c,f]imidazo[1,5-a]azepin-3-amine monohydrobromide 127786-29-2 C16H15N3HBr