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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
5-bromo-2,3-dihydro-1H-inden-1-one 5-溴-2,3-二氢-1H-茚-1-酮 34598-49-7 详细
6-chloro-1H,2H-pyrido[2,3-b]pyrazin-2-one 70395-75-4 详细
2-[(tert-butoxy)carbonyl]-1,2,3,4-tetrahydroisoquinoline-7-carboxylic acid 2-[(叔-丁氧基)羰基]-1,2,3,4-四氢异喹啉-7-羧酸 149353-95-7 详细
3-amino-4-nitro-benzonitrile 3-氨基-4-硝基苯甲腈 99512-10-4 详细
XL-147 956958-53-5 详细
7-bromo-5-fluoro-indan-1-one 1260016-95-2 详细
tert-butyl 3-bromo-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate 叔-丁基 3-溴-4H,5H,6H,7H-吡唑并[1,5-a]吡嗪-5-甲酸基酯 1196154-25-2 详细
tert-butyl N-[(1S)-4-cyano-2,3-dihydro-1H-inden-1-yl]carbamate 叔丁基-N - [(1S)-4-氰基-2,3-二氢-1H-茚-1-基]氨基甲酸 1306763-31-4 详细
2-chloro-6,7-dihydro-5H-pyrrolo[3,4-b]pyridine;hydrochloride 2-氯-5H,6H,7H-吡咯并[3,4-b]吡啶盐酸 1841081-37-5 详细
ethyl 5,5-dimethyl-1H,4H,5H,6H-cyclopenta[b]pyrrole-2-carboxylate 1346674-20-1 详细
tert-butyl 4-benzyloxy-2-methylsulfanyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carboxylate 2648554-48-5 详细
(3S)-6-(trifluoromethyl)-2,3-dihydrobenzofuran-3-amine;hydrochloride 2682097-48-7 详细
6-bromo-2,7-dimethyl-3H-pyrido[2,3-d]pyrimidin-4-one 2090991-89-0 详细
1,2-dihydroquinoxalin-2-one 1196-57-2 详细
tert-butyl 3-amino-6,6-dimethyl-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxylate 叔-丁基 3-氨基-6,6-二甲基-1H,4H,5H,6H-吡咯并[3,4-c]吡唑-5-甲酸基酯 398491-61-7 详细
4,6-dichloropyrido[3,4-d]pyrimidine 4,6-二氯吡啶并[3,4-d]嘧啶 171178-48-6 详细
1-oxo-2,3-dihydro-1H-indene-4-carbonitrile 1-氧亚基-2,3-二氢-1H-茚-4-甲腈 60899-34-5 详细
7-benzyl-2,4-dichloro-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine 7-苯甲基-2,4-二氯-5H,6H,7H,8H-吡啶并[3,4-d]嘧啶 1059735-34-0 详细
4-(tert-butoxycarbonylamino)-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxylic acid 4-{[(叔-丁氧基)羰基]氨基}-1-{7H-吡咯并[2,3-d]嘧啶-4-基}哌啶-4-羧酸 956460-96-1 详细
1-(trifluoromethyl)-3H-1λ3,2-benziodaoxol-3-one TOGNI试剂II 887144-94-7 详细
tert-butyl 7-chloro-3,4-dihydro-2H-1,8-naphthyridine-1-carboxylate 679392-23-5 详细
3-iodo-4,5,6,7-tetrahydro-1H-indazole 3-碘-4,5,6,7-四氢-1H-吲唑 945925-78-0 详细
ethyl cis-2-phenylcyclopropanecarboxylate 946-38-3 详细
6-benzyl-2,4-dichloro-5H,6H,7H,8H-pyrido[4,3-d]pyrimidine 6-苯甲基-2,4-二氯-5H,6H,7H,8H-吡啶并[4,3-d]嘧啶 778574-06-4 详细
2,2-dimethyl-7-tetrahydropyran-2-yloxy-chromene-3-carbaldehyde 1298093-47-6 详细
methyl 3-chloroquinoxaline-6-carboxylate 948833-63-4 详细
7-chloro-4-methyl-2H-pyrido[3,4-d]pyridazin-1-one 2654746-75-3 详细
6-bromo-1,2,3,4-tetrahydroisoquinolin-1-one 6-溴-1,2,3,4-四氢异喹啉-1-酮 147497-32-3 详细
4,7-dichloro-1,6-naphthyridine 952138-13-5 详细
4-Chloro-3-nitrobenzenesulfonamide 4-氯-3-硝基苯磺酰胺 97-09-6 详细
4,6-dichloropyrido[3,2-d]pyrimidine 4,6-二氯吡啶并[3,2-d]嘧啶 175358-02-8 详细
tert-butyl 3-iodo-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxylate 叔-丁基 3-碘-1H,4H,5H,6H,7H-吡唑并[4,3-c]吡啶-5-甲酸基酯 661487-17-8 详细
2,4-dichloro-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine hydrochloride 2,4-二氯-5H,6H,7H,8H-吡啶并[3,4-d]嘧啶盐酸 1187830-76-7 详细
(3R,4S)-1-[(tert-butoxy)carbonyl]-4-phenylpyrrolidine-3-carboxylic acid 956101-09-0 详细
tert-butyl N-[(3S)-6-cyano-2,3-dihydrobenzofuran-3-yl]carbamate 2364560-68-7 详细
benzyl 2,4-dichloro-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carboxylate 1370411-44-1 详细
2,3-Dihydrobenzofuran-4-carbaldehyde 209256-42-8 详细
tert-butyl 3-(tetramethyl-1,3,2-dioxaborolan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate 1798843-08-9 详细
methyl 1,2,3,4-tetrahydroisoquinoline-7-carboxylate hydrochloride 甲基 1,2,3,4-四氢异喹啉-7-甲酸基酯盐酸 220247-69-8 详细
2,4-dichloropyrido[2,3-d]pyrimidine 2,4-二氯吡啶并[2,3-D]嘧啶 126728-20-9 详细
tert-butyl 7-bromo-1,2,3,4-tetrahydroisoquinoline-2-carboxylate 258515-65-0 详细
7-bromo-1H-pyrido[2,3-b]pyrazin-2-one 959616-05-8 详细
2,3-dihydro-1-benzofuran-4-ol 144822-82-2 详细
tert-butyl 4-chloro-5H,6H,7H,8H-pyrido[4,3-d]pyrimidine-6-carboxylate 叔-丁基 4-氯-5H,6H,7H,8H-吡啶并[4,3-d]嘧啶-6-甲酸基酯 1056934-87-2 详细
ethyl 6-chloro-4-oxo-chromene-2-carboxylate 38322-69-9 详细
2,6-difluoro-4-hydroxyphenylboronic acid 957065-87-1 详细
4-[[2-[[(1R,2R)-2-hydroxycyclohexyl]amino]-1,3-benzothiazol-6-yl]oxy]-N-methyl-pyridine-2-carboxamide 953769-46-5 详细
3-(trifluoromethyl)-5H,6H,7H,8H-imidazo[1,5-a]pyrazine 3-(三氟甲基)-5H,6H,7H,8H-咪唑并[1,5-a]吡嗪 959238-29-0 详细
4-chloro-6-methoxy-1,7-naphthyridine 952059-61-9 详细
tert-butyl 4-chloro-2-methyl-5,7-dihydropyrrolo[3,4-d]pyrimidine-6-carboxylate 1393575-79-5 详细
methyl 1,2,3,4-tetrahydroisoquinoline-8-carboxylate hydrochloride 甲基 1,2,3,4-四氢异喹啉-8-甲酸基酯盐酸 1029689-82-4 详细
4-chloro-7,7-difluoro-2-methylsulfanyl-5,6-dihydrocyclopenta[d]pyrimidine 1644414-78-7 详细
2,4,7-trichloro-8-methyl-pyrido[4,3-d]pyrimidine 2454396-72-4 详细
(3R)-6-bromo-2,3-dihydrobenzofuran-3-amine hydrochloride 2703746-10-3 详细
(3S)-6-(trifluoromethyl)-2,3-dihydrofuro[2,3-b]pyridin-3-amine 2382612-91-9 详细
6-bromo-7-methoxy-2-methyl-3H-pyrido[2,3-d]pyrimidin-4-one 2755824-07-6 详细
(2R)-2,3-dihydro-1H-indole-2-carboxylic acid (2R)-2,3-二氢-1H-吲哚-2-羧酸 98167-06-7 详细
tert-butyl 4-chloro-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxylate 叔-丁基 4-氯-5H,6H,7H,8H-吡啶并[3,4-d]嘧啶-7-甲酸基酯 1053656-57-7 详细
5H,7H-furo[3,4-b]pyridine-5,7-dione 5H,7H-呋喃并[3,4-b]吡啶-5,7-二酮 699-98-9 详细
6-bromo-7-methyl-indan-1-one 1071727-49-5 详细
7-bromo-3,3-dimethyl-1,2,3,4-tetrahydroisoquinoline 1338097-15-6 详细
5-bromo-1,2,3,4-tetrahydroquinoline 5-溴-1,2,3,4-四氢喹啉 114744-50-2 详细
7-bromo-3-butyl-8-methoxy-3,5-dihydro-2H-1,5-benzothiazepin-4-one 2649100-07-0 详细
2-iodo-4-methylsulfanyl-7,8-dihydro-6H-quinazolin-5-one 2901099-36-1 详细
2,4-dichloro-5H,7H,8H-pyrano[4,3-d]pyrimidine 2,4-二氯-5H,7H,8H-吡喃并[4,3-d]嘧啶 944902-88-9 详细
(1S)-1-amino-2,3-dihydro-1H-indene-4-carbonitrile hydrochloride 1306763-57-4 详细
tert-butyl 7-(hydroxymethyl)-1,2,3,4-tetrahydroisoquinoline-2-carboxylate 960305-55-9 详细
7-bromo-1,2,3,4-tetrahydroisoquinoline hydrochloride 7-溴-1,2,3,4-四氢异喹啉盐酸 220247-73-4 详细
6-bromo-7-chloro-2-methylsulfanyl-pyrido[2,3-d]pyrimidine 352328-88-2 详细
7-fluoro-2-hydroxy-pyrido[1,2-a]pyrimidin-4-one 1449598-85-9 详细
4-methoxyindan-1-one 13336-31-7 详细
tert-butyl 5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2,3-dihydropyrrolo[2,3-b]pyridine-1-carboxylate 2378821-30-6 详细
hemi(oxalic acid);(5R)-2-(trifluoromethyl)-6,7-dihydro-5H-cyclopenta[b]pyridin-5-amine 2828019-34-5 详细
4-methyl-3-nitro-benzoic acid 96-98-0 详细
7-methoxy-1,4-dihydro-1,6-naphthyridin-4-one 7-甲氧基-1,4-二氢-1,6-萘啶-4-酮 952138-18-0 详细
1,4-dichloro-5H,6H,7H-cyclopenta[d]pyridazine 91846-80-9 详细
6-bromo-2-(methylsulfanyl)-7H,8H-pyrido[2,3-d]pyrimidin-7-one 352328-87-1 详细
tert-butyl 2-chloro-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxylate 叔-丁基 2-氯-5H,6H,7H,8H-吡啶并[3,4-d]嘧啶-7-甲酸基酯 1196156-15-6 详细
2-[(6-chloropyridazin-3-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione 948996-03-0 详细
Vortioxetine hydrobromide 960203-27-4 详细
tert-butyl 3-bromo-5,6,7,8-tetrahydro-1,6-naphthyridine-6-carboxylate 叔-丁基 3-溴-5,6,7,8-四氢-1,6-萘啶-6-甲酸基酯 1184950-48-8 详细
3,5-dihydro-2H-furo[3,2-c]pyridin-4-one 54415-78-0 详细
(3S)-6-bromo-2,3-dihydrobenzofuran-3-amine;hydrochloride 2225878-88-4 详细
7-bromo-2-chloroquinoxaline 7-溴-2-氯喹喔啉 89891-65-6 详细
6-bromo-2,3-dihydro-1H-indole 6-溴吲哚啉 63839-24-7 详细
Rotigotine 99755-59-6 详细
6-chloro-3H-pyrido[3,2-d]pyrimidin-4-one 6-氯-3H,4H-吡啶并[3,2-d]嘧啶-4-酮 171178-33-9 详细
methyl 2-[2-(tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]acetate 甲基 2-[2-(四甲基-1,3,2-二噁硼戊环-2-基)苯基]醋酸盐 956229-86-0 详细
4-(hydroxymethyl)-3-methoxybenzoic acid 4-(羟甲基)-3-甲氧基苯甲酸 955117-56-3 详细
6-chloro-1,2,3,4-tetrahydro-2,7-naphthyridine;hydrochloride 1335053-26-3 详细
3,3-dimethylindan-4-ol 82615-36-9 详细
3-chloro-1-methoxy-5,6-dihydrocyclopenta[c]pyridin-7-one 2747098-69-5 详细
6,8-dichloro-2H-2,7-naphthyridin-1-one 950746-21-1 详细
2-(methylsulfanyl)-7H,8H-pyrido[2,3-d]pyrimidin-7-one 2-(甲基巯基)-7H,8H-吡啶并[2,3-d]嘧啶-7-酮 211244-81-4 详细
arn-509 956104-40-8 详细
4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]aniline 4-[4-(4-甲基哌嗪-1-基)哌啶-1-基]苯胺 959795-70-1 详细
6-bromo-1,2-dihydrophthalazin-1-one 6-溴-1,2-二氢酞嗪-1-酮 75884-70-7 详细
tert-butyl 6-amino-1,1-dimethyl-3,4-dihydroisoquinoline-2-carboxylate 1311134-27-6 详细
1H,3H-furo[3,4-c]pyridine-1,3-dione 1H,3H-呋喃并[3,4-c]吡啶-1,3-二酮 4664-08-8 详细
3-methyl-4,5-dihydrocyclopenta[d]imidazol-6-one 1550999-77-3 详细
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