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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
JQ 1 1268524-70-4 详细
(5R)-5H,6H,7H-cyclopenta[b]pyridin-5-amine 1269843-76-6 详细
methyl isoindoline-4-carboxylate hydrochloride 甲基异二氢吲哚-?4-?甲酸基酯盐酸 127168-90-5 详细
1-[[(2R,3S)-2-(2,4-difluorophenyl)-3-methyl-oxiran-2-yl]methyl]-1,2,4-triazole 127000-90-2 详细
(5S)-6,7-dihydro-5H-cyclopenta[b]pyridin-5-amine 1269934-54-4 详细
SNS-062 1270014-40-8 详细
ethyl 7-bromo-4-chloro-1,5-naphthyridine-3-carboxylate 乙基 7-溴-4-氯-1,5-萘啶-3-甲酸基酯 127448-21-9 详细
(1S,6R,8S)-7,7-dichloro-11,11-dimethyl-5-oxa-3λ-thia-4-azatetracyclo[6.2.1.01,.0,]undecane-3,3-dione 127184-05-8 详细
8-bromo-6-chloro-2-cyclopropylimidazo[1,2-b]pyridazine 1298031-95-4 详细
tert-butyl N-[3-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]oxetan-3-yl]carbamate 1279090-25-3 详细
JNJ-42847922 1293281-49-8 详细
Verteporfin 129497-78-5 详细
4,6-dihydropyrazolo[1,5-c]thiazole-3-carboxylic acid 1286755-08-5 详细
5-tert-butoxycarbonyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-3-carboxylic acid 1280214-48-3 详细
(2S)-2-(trifluoromethyl)oxirane 130025-34-2 详细
3-(2-chloroethyl)-9-hydroxy-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-4-one 130049-77-3 详细
3-(2-{imidazo[1,2-b]pyridazin-3-yl}ethynyl)-4-methylbenzoic acid 3-(2-{咪唑并[1,2-b]哒嗪-3-基}乙炔基)-4-甲基苯甲酸 1300690-48-5 详细
8-chloro-1,7-naphthyridine 8-氯-1,7-萘啶 13058-77-0 详细
8-methoxy-1,2,3,4-tetrahydronaphthalen-1-one 13185-18-7 详细
1-(oxolan-3-yl)-1H-pyrazol-4-amine 1-(噁戊环-3-基)-1H-吡唑-4-胺 1311369-72-8 详细
tert-butyl 3-(chloromethyl)-6,7-dihydro-4H-triazolo[1,5-a]pyrazine-5-carboxylate 1305336-27-9 详细
4-[(3-carboxy-2-hydroxy-1-naphthyl)methyl]-3-hydroxy-naphthalene-2-carboxylic acid 130-85-8 详细
6-chloro-1,4-dihydro-1,5-naphthyridin-4-one 1312760-59-0 详细
tert-butyl (2R)-2-(4-bromophenyl)morpholine-4-carboxylate 1312566-00-9 详细
ABT-494 1310726-60-3 详细
4,7-difluoroindan-1-one 130408-16-1 详细
5-tert-butoxycarbonyl-1-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxylic acid 1306739-66-1 详细
quinoxaline-6-carbaldehyde 130345-50-5 详细
1-(3-cyanophenyl)cyclobutanecarboxylic acid 1314744-75-6 详细
(R)-(6-methoxy-4-quinolyl)-[(1S,2S,4S,5R)-5-vinylquinuclidin-2-yl]methanol 130-95-0 详细
ONO-4059 1351636-18-4 详细
N-{2-[(2S)-2-{5-[(3S)-3-aminopyrrolidin-1-yl]-6-methylpyrazolo[1,5-a]pyrimidin-2-yl}piperidine-1-carbonyl]-4-chlorophenyl}methanesulfonamide 1353625-73-6 详细
2-methyl-2H,3H,5H,6H,7H,8H-pyrido[4,3-c]pyridazin-3-one 1341677-30-2 详细
6-iodo-2-methyl-indan-1-one 1332608-72-6 详细
5-bromo-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzaldehyde 1352819-26-1 详细
3,4,6,7,8,9-hexahydro-2H-pyrazino[1,2-a]indol-1-one 1346672-36-3 详细
1-(oxetan-3-yl)-1H-pyrazol-5-amine 1-(噁丁环烷-3-基)-1H-吡唑-5-胺 1349708-97-9 详细
tert-butyl 4-(oxetan-3-ylamino)piperidine-1-carboxylate 1349718-24-6 详细
6-bromo-8-fluoro-tetralin-2-one 1337857-08-5 详细
2-ethylbutyl (2S)-2-{[(S)-(4-nitrophenoxy)(phenoxy)phosphoryl]amino}propanoate 1354823-36-1 详细
5-bromo-7-fluoro-1,2,3,4-tetrahydronaphthalen-2-one 1336954-16-5 详细
JNJ-42165279 1346528-50-4 详细
tert-butyl 3-(4-bromophenyl)-3-fluoro-azetidine-1-carboxylate 叔-丁基 3-(4-溴苯基)-3-氟吖丁啶-1-甲酸基酯 1357614-51-7 详细
CUDC-907 1339928-25-4 详细
(3S)-3-(4-chlorophenyl)piperidine 1336067-62-9 详细
PyBroP 132705-51-2 详细
5-[(tert-butoxy)carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid 5-[(叔-丁氧基)羰基]-4H,5H,6H,7H,8H-吡唑并[1,5-a][1,4]二氮杂卓-2 1355170-97-6 详细
ethyl trans-2-(4-cyanophenyl)cyclopropanecarboxylate 132145-60-9 详细
6,7-dihydro-5H-pyrrolo[3,4-b]pyridine-3-carbonitrile;hydrochloride 1346808-69-2 详细
tert-butyl 3-(cyclopropylamino)azetidine-1-carboxylate 1342433-96-8 详细
2-(3-methoxyphenyl)-1-piperazin-1-yl-ethanone;hydrochloride 1356998-47-4 详细
2-methyl-5,6,7,8-tetrahydro-3H-pyrido[4,3-d]pyrimidin-4-one 134201-14-2 详细
4,4-dimethyl-1,10-diazatricyclo[6.4.0.02,]dodeca-2(6),7-dien-9-one 1346674-23-4 详细
3-fluoro-5H,6H,7H-pyrrolo[3,4-b]pyridine hydrochloride 3-氟-5H,6H,7H-吡咯并[3,4-b]吡啶盐酸 1346808-65-8 详细
Olmutinib 奥姆替尼 1353550-13-6 详细
tert-butyl 3-(6-amino-3-pyridyl)azetidine-1-carboxylate 1346673-86-6 详细
N-(6-azaspiro[2.5]octan-2-ylmethyl)-N-methyl-cyclopropanamine 1339505-47-3 详细
propan-2-yl (2S)-2-{[(S)-pentafluorophenoxy(phenoxy)phosphoryl]amino}propanoate N-[(S)-(2,3,4,5,6-五氟苯氧基)苯氧基磷酰基]-L-丙氨酸异丙酯 1334513-02-8 详细
2-amino-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzaldehyde 2-氨基-5-(四甲基-1,3,2-二噁硼戊环-2-基)苯(甲)醛 1319197-32-4 详细
cis-3-fluoro-1-(3-fluoropyridin-2-yl)cyclobutane-1-carbonitrile 顺-3-氟-1-(3-氟吡啶-2-基)环丁烷-1-甲腈 1344145-38-5 详细
ethyl 1-oxo-3,4-dihydro-2H-pyrrolo[1,2-a]pyrazine-7-carboxylate 1338563-13-5 详细
8-bromo-6-methoxy-tetralin-1-one 1336952-02-3 详细
2-isopropoxy-5-methyl-4-(4-piperidyl)aniline;dihydrochloride 5-甲基-4-(哌啶-4-基)-2-(丙烷-2-氧基)苯胺二盐酸 1380575-45-0 详细
3-(4-chlorophenyl)cyclobutane-1-carboxylic acid 1384429-60-0 详细
6,7-difluorotetralin-1-one 137114-68-2 详细
3-(3-bromophenyl)oxetan-3-ol 3-(3-溴苯基)噁丁环烷-3-醇 1379811-98-9 详细
3-(3-bromophenyl)oxetane-3-carboxylic acid 1363381-80-9 详细
2-[4-(bromomethyl)phenyl]-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2-[4-(溴甲基)苯基]-4,4,5,5-四甲基-1,3,2-二噁硼戊环 138500-85-3 详细
6-(1-methyl-4-piperidyl)pyridin-3-amine 1373421-18-1 详细
6-methoxyindan-1-one 13623-25-1 详细
4-[(2S)-pyrrolidin-2-yl]benzoic acid;hydrochloride 1381927-91-8 详细
PRT 062607 1370261-98-5 详细
3-[(3,5-dimethoxyphenyl)methyl]azetidine hydrochloride 1376321-05-9 详细
2-(1,3,2-benzodioxaborol-2-yl)-1,3,2-benzodioxaborole 13826-27-2 详细
3-(3-bromophenyl)oxetan-3-yl]methanol 1363382-09-5 详细
cerdulatinib hydrochloride 1369761-01-2 详细
tert-butyl (2R)-2-(4-bromo-1H-imidazol-2-yl)pyrrolidine-1-carboxylate 叔-丁基 (2R)-2-(4-溴-1H-咪唑-2-基)吡咯烷-1-甲酸基酯 1370600-56-8 详细
2-bromo-6,7-dihydro-5H-furo[3,2-c]pyridin-4-one 1379361-49-5 详细
2-azatricyclo[10.4.0.0]hexadeca-1(12),4(9),5,7,13,15-hexaen-10-yne 1369862-03-2 详细
4-chloro-5H,6H,7H-pyrrolo[3,4-d]pyrimidine hydrochloride 4-氯-5H,6H,7H-吡咯并[3,4-d]嘧啶盐酸 1373228-90-0 详细
2-[(8R)-8-(3,5-difluorophenyl)-8-methyl-10-oxo-6,9-diazaspiro[4.5]decan-9-yl]-N-[(6S)-2'-oxo-1',2',5,7-tetrahydrospiro[cyclopenta[b]pyridine-6,3'-pyrrolo[2,3-b]pyridin]-3-yl]acetamide 1380887-60-4 详细
(1S)-1-[3-(difluoromethyl)-2-fluoro-phenyl]ethanamine 1389366-49-7 详细
3-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine;hydrochloride 1358784-11-8 详细
Elbasvir 1370468-36-2 详细
6-bromo-3,4-dihydro-2H-pyrrolo[1,2-a]pyrazin-1-one 1374684-64-6 详细
1-(4-fluorophenyl)-1H-pyrazole-4-carboxylic acid 138907-81-0 详细
2-[(tert-butoxy)carbonyl]-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-6-carboxylic acid 2-[(叔-丁氧基)羰基]-1H,2H,3H,4H-吡咯并[1,2-a]吡嗪-6-羧酸 1363380-86-2 详细
7-bromo-2,3,4,5-tetrahydro-1,4-benzoxazepine-5-carboxylic acid 1378254-82-0 详细
4-(3-piperidyl)oxazole 1367989-82-9 详细
3-(4-chlorophenyl)oxetane-3-carboxylic acid 3-(4-氯苯基)噁丁环烷-3-羧酸 1393534-20-7 详细
7-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-one 7-(三氟甲基)-1,2,3,4-四氢异喹啉-1-酮 1365759-12-1 详细
1-methyl-4-{2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]ethyl}piperazine 1-甲基-4-{2-[4-(4,4,5,5-四甲基-1,3,2-二噁硼戊环-2-基)-1H-吡唑-1-基]乙基}哌嗪 1392419-83-8 详细
(3S)-6-fluoro-1,2,3,4-tetrahydroisoquinolin-3-yl]methanol 1389391-15-4 详细
3-(2-chloropyrimidin-5-yl)-5,5-dimethyl-imidazolidine-2,4-dione 1380698-64-5 详细
6'-bromo-1',2'-dihydrospiro[cyclopropane-1,3'-indole 1379360-39-0 详细
4-bromo-1H,2H,3H-pyrrolo[2,3-b]pyridine 4-溴-1H,2H,3H-吡咯并[2,3-b]吡啶 1393534-35-4 详细
6-(4-bromophenyl)morpholin-3-one 1368418-27-2 详细
5-tert-butyl 3-ethyl 4H,5H,6H,7H-thieno[3,2-c]pyridine-3,5-dicarboxylate 5-叔-丁基 3-乙基 4H,5H,6H,7H-噻吩并[3,2-c]吡啶-3,5-二甲酸基酯 1363381-39-8 详细
3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazine 1383675-83-9 详细
3-(2,4-difluorophenyl)azetidin-3-ol 1388073-15-1 详细
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