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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
5H,6H,7H,8H-imidazo[1,5-a]pyrazine 5H,6H,7H,8H-咪唑并[1,5-a]吡嗪 297172-19-1 详细
6-bromo-1-chlorophthalazine 6-溴-1-氯酞嗪 470484-70-9 详细
5-bromo-1,3-dihydro-benzo(c)thiophene 2,2-dioxide 5-溴-1,3-二氢-苯并(c)噻吩 2,2-二氧化 351005-12-4 详细
2-bromo-5-methyl-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridine 2-溴-5-甲基-4H,5H,6H,7H-[1,3]噻唑并[5,4-c]吡啶 143150-92-9 详细
3,3-dimethyl-2,3-dihydro-1H-indole 3,3-二甲基-2,3-二氢-1H-吲哚 1914-02-9 详细
methyl 5-bromo-2,3-dihydro-1h-indole-6-carboxylate 甲基 5-溴-2,3-二氢-1h-吲哚-6-甲酸基酯 1788041-64-4 详细
6-chloro-1,2,3,4-tetrahydroisoquinolin-1-one 6-氯-1,2,3,4-四氢异喹啉-1-酮 22246-02-2 详细
6-bromophthalazine 6-溴酞嗪 19064-74-5 详细
4-oxo-3,4-dihydrophthalazine-1-carboxylic acid 3260-44-4 详细
indan-4-amine 32202-61-2 详细
methyl isoindoline-5-carboxylate;hydrochloride 2,3-二氢-1H-异吲哚-5-羧酸甲酯盐酸 127168-93-8 详细
tert-butyl 2-chloro-5,7-dihydropyrrolo[3,4-d]pyrimidine-6-carboxylate 2-氯-5H,6H,7H-吡咯并[3,4-d]嘧啶-6-甲酸叔丁酯 1211581-47-3 详细
3-bromo-6,7-dihydrocyclopenta[b]pyridin-5-one 1196154-87-6 详细
2,4-dichloro-5H,7H-thieno[3,4-d]pyrimidine 2,4-二氯-5H,7H-噻吩并[3,4-d]嘧啶 74901-71-6 详细
tert-butyl 4-hydroxy-2,3-dihydro-1H-isoindole-2-carboxylate 叔-丁基 4-羟基-2,3-二氢-1H-异吲哚-2-甲酸基酯 871013-92-2 详细
2-chloro-5H,6H,7H-pyrrolo[3,4-d]pyrimidine hydrochloride 2-氯-5H,6H,7H-吡咯并[3,4-d]嘧啶盐酸 1314790-85-6 详细
3H,4H-pyrido[2,3-d]pyrimidin-4-one 3H,4H-吡啶并[2,3-d]嘧啶-4-酮 24410-19-3 详细
2,4,7-trichloro-8-methoxy-pyrido[4,3-d]pyrimidine 2454491-03-1 详细
7-bromo-1,2,3,4-tetrahydroquinoline 7-溴-1,2,3,4-四氢喹啉 114744-51-3 详细
2,2,4-trimethyl-1H-quinolin-6-ol 72107-05-2 详细
5-methyl-6,7-dihydro-4H-thiazolo[4,5-c]pyridin-2-amine 5-甲基-4H,5H,6H,7H-[1,3]噻唑并[4,5-c]吡啶-2-胺 784079-98-7 详细
1,4-dichloropyrido[3,4-d]pyridazine 14490-19-8 详细
2,3-dihydro-1H-pyrrolo[3,2-c]pyridine 23596-28-3 详细
1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-one 1H,4H,5H,6H,7H-吡咯并[3,2-c]吡啶-4-酮 736990-65-1 详细
1,3-dimethyl-5,6-dihydro-4H-pyrrolo[3,4-c]pyrazole;dihydrochloride 2753455-95-5 详细
tert-butyl 5-bromo-2,3-dihydro-1H-isoindole-2-carboxylate 201940-08-1 详细
2,4-dichloro-5H,6H,7H-cyclopenta[d]pyrimidine 5466-43-3 详细
4,5,6,7-tetrahydro-1H-indole 4,5,6,7-四氢-1H-吲哚 13618-91-2 详细
tert-butyl 3-iodo-1H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridine-6-carboxylate 1638765-22-6 详细
1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine 1H,2H,3H,4H-吡咯并[1,2-a]吡嗪 71257-38-0 详细
methyl indoline-5-carboxylate 2,3-二氢-1H-吲哚-5-羧酸甲酯 141452-01-9 详细
6-chloro-1-(p-tolylsulfonyl)-2,3-dihydroquinolin-4-one 857762-10-8 详细
7-bromo-3,4-dihydro-1H-2-benzopyran-4-one 168759-64-6 详细
7-methoxy-1-methyl-tetralin-2-one 1204-23-5 详细
ethyl 5,6,7,8-tetrahydroimidazo[1,2-a]pyrazine-2-carboxylate hydrochloride 623906-17-2 详细
5H,7H-furo[3,4-b]pyrazine-5,7-dione 4744-50-7 详细
2-methyl-1,2,3,4-tetrahydroisoquinolin-7-amine 2-甲基-1,2,3,4-四氢异喹啉-7-胺 14097-40-6 详细
6-bromo-2,3-dihydro-1H-1,8-naphthyridin-4-one 676515-34-7 详细
ethyl 6-hydroxy-1,2,3,4-tetrahydroisoquinoline-3-carboxylate hydrochloride 乙基 6-羟基-1,2,3,4-四氢异喹啉-3-甲酸基酯盐酸 128073-39-2 详细
5-fluoro-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one 5-氟-1,2,3,4-四氢-1,8-萘啶-2-酮 1237535-78-2 详细
2,4,8-trichloropyrido[3,4-d]pyrimidine 1470249-17-2 详细
1,2,3,4-tetrahydroisoquinolin-6-ol 1,2,3,4-四氢异喹啉-6-酚 14446-24-3 详细
methyl 8-hydroxy-2-[(4-methoxyphenyl)methyl]-1-oxo-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate 2306268-97-1 详细
4,5,6,7-tetrahydro-1-benzothiophen-4-one 13414-95-4 详细
tert-butyl 6-bromo-1,2,3,4-tetrahydroisoquinoline-2-carboxylate 893566-74-0 详细
4-bromo-2,3-dihydro-1H-isoindole hydrochloride 4-溴-2,3-二氢-1H-异吲哚盐酸 923590-95-8 详细
6-bromo-3H,4H-pyrido[2,3-d]pyrimidin-4-one 6-溴-3H,4H-吡啶并[2,3-d]嘧啶-4-酮 155690-79-2 详细
4-bromo-1H,2H,3H-pyrrolo[2,3-c]pyridine 4-溴-1H,2H,3H-吡咯并[2,3-c]吡啶 1617514-93-8 详细
2-bromo-6,7-dihydro-5H-pyrazolo[1,5-a]pyrazin-4-one 2468022-89-9 详细
4-chloropyrido[3,2-d]pyrimidine 4-氯吡啶并[3,2-d]嘧啶 51674-77-2 详细
4H,5H,6H,7H-pyrazolo[1,5-a]pyrimidine 4H,5H,6H,7H-吡唑并[1,5-a]嘧啶 126352-69-0 详细
1,2,3,4-tetrahydroquinolin-3-ol 1,2,3,4-四氢喹啉-3-酚 3418-45-9 详细
(2R)-2-methyl-2,3-dihydro-1H-indole (2R)-2-甲基-2,3-二氢-1H-吲哚 22160-13-0 详细
5-bromo-2,3-dihydro-1H-isoindole hydrochloride 5-溴-2,3-二氢-1H-异吲哚盐酸 919346-89-7 详细
2,4,7-trichloropyrido[2,3-d]pyrimidine 2,4,7-三氯吡啶并[2,3-d]嘧啶 938443-20-0 详细
7-chloro-2-(methylsulfanyl)pyrido[2,3-d]pyrimidine 352328-41-7 详细
benzyl 2,4-dichloro-5h,6h,7h,8h-pyrido[4,3-d]pyrimidine-6-carboxylate 苯甲基 2,4-二氯-5h,6h,7h,8h-吡啶并[4,3-d]嘧啶-6-甲酸基酯 1160248-14-5 详细
3-chloro-1,2-dihydroquinoxalin-2-one 3-氯-1,2-二氢喹喔啉-2-酮 35676-70-1 详细
7-methoxy-1,2,3,4-tetrahydroisoquinolin-1-one 7-甲氧基-1,2,3,4-四氢异喹啉-1-酮 22246-04-4 详细
6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidine-2,4-diol;2,2,2-trifluoroacetic acid 2387597-16-0 详细
4H,5H,6H,7H-thieno[3,2-c]pyridine,hydrochloride 4H,5H,6H,7H-噻吩并[3,2-c]吡啶,盐酸 28783-41-7 详细
5H,6H,7H-cyclopenta[c]pyridin-5-one 5H,6H,7H-环戊二烯并[c]吡啶-5-酮 350847-80-2 详细
5-bromo-1,2,3,4-tetrahydroisoquinoline hydrochloride 5-溴-1,2,3,4-四氢异喹啉盐酸 923591-51-9 详细
tert-butyl 5-hydroxy-3,4-dihydro-1H-isoquinoline-2-carboxylate 216064-48-1 详细
6-bromo-2,4-dichloropyrido[2,3-d]pyrimidine 6-溴-2,4-二氯吡啶并[2,3-d]嘧啶 1234616-70-6 详细
3-bromo-6,7-dihydro-4H-pyrazolo[5,1-c][1,4]oxazine 1393558-10-5 详细
4-chloro-2,3-dihydro-1H-pyrrolo[2,3-b]pyridine;hydrochloride 4-氯-1H,2H,3H-吡咯并[2,3-b]吡啶盐酸 1818847-83-4 详细
8-chloro-2-methylsulfonyl-pyrido[3,4-d]pyrimidine 1578246-63-5 详细
2-(trifluoromethyl)-6,7-dihydrocyclopenta[b]pyridin-5-one 1196155-83-5 详细
4,7-dichloro-8-fluoro-pyrido[4,3-d]pyrimidine 2454396-94-0 详细
6-bromo-4-chlorocinnoline 6-溴-4-氯曾嗪 68211-15-4 详细
8-bromo-2-chloroquinoxaline 1092500-67-8 详细
ethyl 4,5,6,7-tetrahydro-1H-indole-2-carboxylate 65880-18-4 详细
1,5,6,7-tetrahydroindazol-4-one 499206-33-6 详细
6,7-dihydro-5H-pyrrolo[3,4-b]pyridine hydrochloride 651558-51-9 详细
2-chloro-5H,6H,7H,8H-pyrido[4,3-d]pyrimidine hydrochloride 2-氯-5H,6H,7H,8H-吡啶并[4,3-d]嘧啶盐酸 1314723-39-1 详细
3-bromo-5H,7H-furo[3,4-b]pyridine-5,7-dione 3-溴-5H,7H-呋喃并[3,4-b]吡啶-5,7-二酮 98278-78-5 详细
4,5,6,7-tetrahydro-1H-indol-4-one 4,5,6,7-四氢-1H-吲哚-4-酮 13754-86-4 详细
7-bromo-3H,4H-pyrido[3,4-d]pyridazin-4-one 7-溴3H,4H-吡啶并[3,4-d]哒嗪-4-酮 794591-77-8 详细
3-bromo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridine;hydrochloride 3-溴-5H,6H,7H-吡咯并[3,4-b]吡啶盐酸 1394117-24-8 详细
2,3-dihydro-1H-isoindol-5-ol hydrobromide 2,3-二氢-1H-异吲哚-5-酚氢溴酸盐 105358-58-5 详细
2-amino-4,5,6,7-tetrahydro-1,3-benzothiazol-7-one 2-氨基-4,5,6,7-四氢-1,3-苯并噻唑-7-酮 17583-10-7 详细
4,7-dichloro-8-fluoro-2-methyl-pyrido[4,3-d]pyrimidine 2454397-79-4 详细
methyl 2-[(1R)-6-hydroxyindan-1-yl]acetate 1187197-92-7 详细
tert-butyl 2-bromo-4H,5H,6H,7H-thieno[2,3-c]pyridine-6-carboxylate 叔-丁基 2-溴-4H,5H,6H,7H-噻吩并[2,3-c]吡啶-6-甲酸基酯 910443-31-1 详细
2-sulfanylidene-1h,2h,3h,4h-pyrido[3,4-d]pyrimidin-4-one 2-硫烷亚基-1h,2h,3h,4h-吡啶并[3,4-d]嘧啶-4-酮 412341-42-5 详细
tert-butyl 4-bromo-2,3-dihydro-1H-isoindole-2-carboxylate 叔-丁基 4-溴-2,3-二氢-1H-异吲哚-2-甲酸基酯 1035235-27-8 详细
8-bromo-1,2,3,4-tetrahydronaphthalen-1-one 8-溴-1,2,3,4-四氢萘-1-酮 651735-60-3 详细
ethyl 3-bromo-6,6-difluoro-5,7-dihydropyrazolo[5,1-b][1,3]oxazine-2-carboxylate 2128657-45-2 详细
6-[(tert-butoxy)carbonyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridine-3-carboxylic acid 821785-76-6 详细
6-hydroxy-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid 6-羟基-1,2,3,4-四氢异喹啉-3-羧酸 76824-99-2 详细
ethyl 5,6,7,8-tetrahydro-1,7-naphthyridine-3-carboxylate hydrochloride 乙基 5,6,7,8-四氢-1,7-萘啶-3-甲酸基酯盐酸 1207175-08-3 详细
tert-butyl 6-formyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carboxylate 叔-丁基 6-甲酰基-1H,2H,3H,4H-吡咯并[1,2-a]吡嗪-2-甲酸基酯 1174068-79-1 详细
tert-butyl 3-amino-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxylate 叔-丁基 3-氨基-1H,4H,5H,6H,7H-吡唑并[4,3-c]吡啶-5-甲酸基酯 398491-64-0 详细
6-bromo-1,4-dichlorophthalazine 6-溴-1,4-二氯酞嗪 240400-95-7 详细
ethyl 5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate hydrochloride 1384080-92-5 详细
tert-butyl 3-bromo-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxylate 1936429-06-9 详细
tert-butyl 4,6,7,8-tetrahydro-2H-pyrazolo[4,3-c]azepine-5-carboxylate 1935900-29-0 详细
4-bromo-6,7-dihydro-5H-isoquinolin-8-one 1428651-86-8 详细
2-chloro-5,5-dimethyl-5H,6H,7H-pyrrolo[2,3-d]pyrimidine 2-氯-5,5-二甲基-5H,6H,7H-吡咯并[2,3-d]嘧啶 1679381-63-5 详细
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