ERK Inhibitor
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- $32 - $228
- Product name: ERK Inhibitor
- CAS: 1049738-54-6
- MF: C14H17ClN2O3S
- MW: 328.81
- EINECS:
- MDL Number:MFCD09038681
- Synonyms:(5Z)-3-(2-aminoethyl)-5-[(4-ethoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione:hydrochloride;ERK Inhibitor - CAS 1049738-54-6 - Calbiochem;3-(2-aminoethyl)-5-[(4-ethoxyphenyl)methylene]-2,4-thiazolidinedione,monohydrochloride;ERK-IN-4
5 prices
Selected condition：
Brand
- AK Scientific
- Cayman Chemical
- Sigma-Aldrich
Package
- 500μg
- 1mg
- 5mg
- 1 unit
- ManufacturerAK Scientific
- Product number9473CW
- Product descriptionErkInhibitor
- Packaging5mg
- Price$228
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number15944
- Product descriptionERK Inhibitor ≥95%
- Packaging500μg
- Price$32
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number15944
- Product descriptionERK Inhibitor ≥95%
- Packaging1mg
- Price$50
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number15944
- Product descriptionERK Inhibitor ≥95%
- Packaging5mg
- Price$117
- Updated2024-03-01
- Buy
- ManufacturerSigma-Aldrich
- Product number328006-M
- Product descriptionERK Inhibitor The ERK Inhibitor, also referenced under CAS 1049738-54-6, controls the biological activity of ERK. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applica
- Packaging1 unit
- Price$133
- Updated2025-07-31
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | 9473CW | ErkInhibitor | 5mg | $228 | 2021-12-16 | Buy |
| Cayman Chemical | 15944 | ERK Inhibitor ≥95% | 500μg | $32 | 2024-03-01 | Buy |
| Cayman Chemical | 15944 | ERK Inhibitor ≥95% | 1mg | $50 | 2024-03-01 | Buy |
| Cayman Chemical | 15944 | ERK Inhibitor ≥95% | 5mg | $117 | 2024-03-01 | Buy |
| Sigma-Aldrich | 328006-M | ERK Inhibitor The ERK Inhibitor, also referenced under CAS 1049738-54-6, controls the biological activity of ERK. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applica | 1 unit | $133 | 2025-07-31 | Buy |
Properties
storage temp. :+2C to +8C
solubility :DMSO: 2 mg/ml
form :Light yellow solid
color :Off-white to yellow
solubility :DMSO: 2 mg/ml
form :Light yellow solid
color :Off-white to yellow
Safety Information
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Description
ERK inhibitor is a cell-permeable inhibitor that binds ERK2 near its docking domain (KD = 5 μM). This prevents its interaction with protein substrates without inhibiting catalytic activity. ERK inhibitor blocks ERK-specific phosphorylation of ribosomal S6 kinase-1 and ternary complex factor Elk-1 but does not affect ERK1/2 phosphorylation by MEK1/2. Presumably through its effects on ERK, ERK inhibitor completely prevents proliferation of HeLa cells (IC50 = 15-20 μM), A549 lung carcinoma cells (IC50 = 25 μM), Sum-159 estrogen receptor-negative breast cancer cells and HT1080 fibrosarcoma cells.More related product prices
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Suppliers and manufacturers
Shaanxi Cuikang Pharmaceutical Technology Co., Ltd
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Shaanxi Cuikang Pharmaceutical Technology Co., Ltd
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ComMedX (Computational Medicine Beijing Co., Ltd.)
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Sigma-Aldrich
BOC Sciences
