Inhibitor Activator

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Structure Chemical Name CAS MF
BTdCPU BTdCPU 1257423-87-2 C13H8Cl2N4OS
Pyridazine, 3-[[(2-chloro-6-fluorophenyl)methyl]thio]-6-(2-pyridinyl)- Pyridazine, 3-[[(2-chloro-6-fluorophenyl)methyl]thio]-6-(2-pyridinyl)- 892415-28-0 C16H11ClFN3S
[oxido-(2,3,4,5,6-pentaphosphonatooxycyclohexyl)oxyphosphoryl] phosphate [oxido-(2,3,4,5,6-pentaphosphonatooxycyclohexyl)oxyphosphoryl] phosphate 193743-89-4
EG-011 EG-011 2377113-41-0 C28H26N4O4
(1E,4E)-1,5-Bis(2-Methoxyphenyl)penta-1,4-dien-3-one (1E,4E)-1,5-Bis(2-Methoxyphenyl)penta-1,4-dien-3-one 39777-61-2 C19H18O3
WS3 (IΚB/IKK inhibitor) WS3 (IΚB/IKK inhibitor)
PND-1186 (FAK inhibitor) PND-1186 (FAK inhibitor)
PI-103 (PI3K inhibitor) PI-103 (PI3K inhibitor)
PFI-4 (EPIGENETIC READER DOMAIN inhibitor) PFI-4 (EPIGENETIC READER DOMAIN inhibitor)
PANOBINOSTAT (LBH589) (HDAC inhibitor) PANOBINOSTAT (LBH589) (HDAC inhibitor)
OSELTAMIVIR ACID (NEURAMINIDASE Inhibitor) OSELTAMIVIR ACID (NEURAMINIDASE Inhibitor)
NU-7441 (DNA-PK inhibitor) NU-7441 (DNA-PK inhibitor)
MG-132 (PROTEASOME Inhibitor) MG-132 (PROTEASOME Inhibitor)
MASITINIB (C-KIT inhibitor) MASITINIB (C-KIT inhibitor)
IXAZEOMIB (MLN2238) (20S PROTEASOME Inhibitor) IXAZEOMIB (MLN2238) (20S PROTEASOME Inhibitor)
ICOTINIB HCL (EGFR inhibitor) ICOTINIB HCL (EGFR inhibitor)
HYDROXYLAMINE HYDROCHLORIDE/Hydroxylamine Hydrochloride HYDROXYLAMINE HYDROCHLORIDE/Hydroxylamine Hydrochloride Cl2H8N2O2
EPOTHILONE B (MICROTUBULE ASSOSIATED inhibitor) EPOTHILONE B (MICROTUBULE ASSOSIATED inhibitor)
WH-4-023 (SRC inhibitor) WH-4-023 (SRC inhibitor)
TG101348 (JAK inhibitor) TG101348 (JAK inhibitor)
PFI-3 (EPIGENETIC READER DOMAIN inhibitor) PFI-3 (EPIGENETIC READER DOMAIN inhibitor)
PD184352 (MEK inhibitor) PD184352 (MEK inhibitor)
ML324 (HISTONE DEMETHYLASE inhibitor) ML324 (HISTONE DEMETHYLASE inhibitor)
KU0063794 (MTOR inhibitor) KU0063794 (MTOR inhibitor)
JNJ-7777120 (HISTAMINE RECEPTOR antagonist) JNJ-7777120 (HISTAMINE RECEPTOR antagonist)
GSK1292263 (GPR agonist) GSK1292263 (GPR agonist)
BYL719 (PI3K inhibitor) BYL719 (PI3K inhibitor)
BML-210 (HDAC inhibitor) BML-210 (HDAC inhibitor)
2H-Pyran-4-propanamide, α-[4-(cyclopropylsulfonyl)phenyl]-N-(5-fluoro-2-thiazolyl)tetrahydro-, (αR)- 2H-Pyran-4-propanamide, α-[4-(cyclopropylsulfonyl)phenyl]-N-(5-fluoro-2-thiazolyl)tetrahydro-, (αR)- 745051-61-0 C20H23FN2O4S2
VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor) VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor)
U-104 (Carbonic anhydrase inhibitor) U-104 (Carbonic anhydrase inhibitor)
E-64 (CYSTEINE PROTEASE inhibitor) E-64 (CYSTEINE PROTEASE inhibitor)
DOCETAXEL (MICROTUBULE ASSOSIATED inhibitor) DOCETAXEL (MICROTUBULE ASSOSIATED inhibitor)
DEGRASYN (BCR-ABL inhibitor) DEGRASYN (BCR-ABL inhibitor)
CC-223 (MTOR inhibitor) CC-223 (MTOR inhibitor)
BI2536 (PLK inhibitor) BI2536 (PLK inhibitor)
A83-01 (ALK5 inhibitor) A83-01 (ALK5 inhibitor)
A-366 (HISTONE METHYLTRANSFERASE Inhibitor) A-366 (HISTONE METHYLTRANSFERASE Inhibitor)
ICA 069673 ICA 069673 582323-16-8 C11H6ClF2N3O
VOLASERTIB (PLK inhibitor) VOLASERTIB (PLK inhibitor)
TUBASTATIN A (HDAC inhibitor) TUBASTATIN A (HDAC inhibitor)
TEDIZOLID (MAO-A inhibitor) TEDIZOLID (MAO-A inhibitor)
SP600125 (JNK inhibitor) SP600125 (JNK inhibitor)
SB203580 (P38 MAPK Inhibitor) SB203580 (P38 MAPK Inhibitor)
SALIRASIB (RHO inhibitor) SALIRASIB (RHO inhibitor)
RG108 (DNA METHYLTRANSFERASE inhibitor) RG108 (DNA METHYLTRANSFERASE inhibitor)
PLERIXAFOR (CXCR inhibitor) PLERIXAFOR (CXCR inhibitor)
PD-173955 (BCR-ABL inhibitor) PD-173955 (BCR-ABL inhibitor)
ODANACATIB (CYSTEINE PROTEASE inhibitor) ODANACATIB (CYSTEINE PROTEASE inhibitor)
MI-2 (HISTONE METHYLTRANSFERASE Inhibitor) MI-2 (HISTONE METHYLTRANSFERASE Inhibitor)
GSK1278863 (HIF inhibitor) GSK1278863 (HIF inhibitor)
DACOMITINIB (EGFR inhibitor) DACOMITINIB (EGFR inhibitor)
BATIMASTAT (MMP inhibitor) BATIMASTAT (MMP inhibitor)
AVASIMIBE (P450 inhibitor) AVASIMIBE (P450 inhibitor)
SALUBRINAL (PERK inhibitor) SALUBRINAL (PERK inhibitor)
FLAVOPIRIDOL HCL (CDK inhibitor) FLAVOPIRIDOL HCL (CDK inhibitor)
DEFACTINIB (FAK inhibitor) DEFACTINIB (FAK inhibitor)
CEDIRANIB (VEGFR inhibitor) CEDIRANIB (VEGFR inhibitor)
BAY11-7082 (IΚB/IKK inhibitor) BAY11-7082 (IΚB/IKK inhibitor)
(-)-BLEBBISTATIN (ATPASE inhibitor) (-)-BLEBBISTATIN (ATPASE inhibitor)
AG14361 (PARP1 inhibitor) AG14361 (PARP1 inhibitor)
ACP-196 (BTK inhibitor) ACP-196 (BTK inhibitor)
ABT-737 (BCL-2 inhibitor) ABT-737 (BCL-2 inhibitor)
CK-2127107 CK-2127107 1345410-31-2 C19H18F2N6O
VILAZODONE (SSRI inhibitor) VILAZODONE (SSRI inhibitor)
TBA-354 (anti-tuberculosis) TBA-354 (anti-tuberculosis)
SAG (HEDGEHOG/SMOOTHENED agonist) SAG (HEDGEHOG/SMOOTHENED agonist)
PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor) PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor)
OSU-03012 (PDK-1 inhibitor) OSU-03012 (PDK-1 inhibitor)
MONOMETHYL AURISTATIN E (microtubule-associated inhibitor) MONOMETHYL AURISTATIN E (microtubule-associated inhibitor)
ML141 (RHO inhibitor) ML141 (RHO inhibitor)
KN-93 PHOSPHATE (CAMK Inhibitor) KN-93 PHOSPHATE (CAMK Inhibitor)
GSK126 (EZH2 inhibitor) GSK126 (EZH2 inhibitor)
GELDANAMYCIN (HSP90 inhibitor) GELDANAMYCIN (HSP90 inhibitor)
GANT61 (HEDGEHOG/SMOOTHENED Inhibitor) GANT61 (HEDGEHOG/SMOOTHENED Inhibitor)
EPZ-6438 (E7438) (EZH2 inhibitor) EPZ-6438 (E7438) (EZH2 inhibitor)
EMPAGLIFLOZIN (SGLT inhibitor) EMPAGLIFLOZIN (SGLT inhibitor)
DOXORUBICIN (TOPOISOMERASE inhibitor) DOXORUBICIN (TOPOISOMERASE inhibitor)
DAPT (Γ-SECRETASE inhibitor) DAPT (Γ-SECRETASE inhibitor)
DACLATASVIR (HCV NS5A inhibitor) DACLATASVIR (HCV NS5A inhibitor)
COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor) COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor)
CABOZANTINIB (VEGFR inhibitor) CABOZANTINIB (VEGFR inhibitor)
BREFELDIN A (protein transport inhibitor) BREFELDIN A (protein transport inhibitor)
BKM120 (PI3K inhibitor) BKM120 (PI3K inhibitor)
AKT INHIBITOR VIII (AKT inhibitor) AKT INHIBITOR VIII (AKT inhibitor)
ABT-199 (BCL-2 inhibitor) ABT-199 (BCL-2 inhibitor)
Porfiromycin Porfiromycin 801-52-5 C16H20N4O5
VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor) VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor)
TETRABENAZINE (VMAT-2 Inhibitor) TETRABENAZINE (VMAT-2 Inhibitor)
SNX-2112 (PF-04928473) (HSP90 antimony inhibitor) SNX-2112 (PF-04928473) (HSP90 antimony inhibitor)
PLX4032 (RAF inhibitor) PLX4032 (RAF inhibitor)
PD123319 (RAAS inhibitor) PD123319 (RAAS inhibitor)
NS-2028 (SGC inhibitor) NS-2028 (SGC inhibitor)
NECROSTATIN-1 (TNF-ALPHA inhibitor) NECROSTATIN-1 (TNF-ALPHA inhibitor)
ML323 (DUB inhibitor) ML323 (DUB inhibitor)
KU-55933 (ATM inhibitor) KU-55933 (ATM inhibitor)
(+)-JQ1 (BRD4 inhibitor) (+)-JQ1 (BRD4 inhibitor)
GSK2141795 (AKT inhibitor) GSK2141795 (AKT inhibitor)
GANETESPIB (HSP inhibitor) GANETESPIB (HSP inhibitor)
ENZALUTAMIDE (MDV3100) (AR inhibitor) ENZALUTAMIDE (MDV3100) (AR inhibitor)
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