Thalidomide-O-amido-PEG4-C2-NH2 hydrochloride

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Thalidomide-O-amido-PEG4-C2-NH2 hydrochloride manufacturers

Thalidomide-O-amido-PEG4-C2-NH2 hydrochloride Basic information
Product Name:Thalidomide-O-amido-PEG4-C2-NH2 hydrochloride
Synonyms:Thalidomide-O-amido-PEG4-C2-NH2 hydrochloride;-oxyacetamide-PEG4-amine;N-(14-Amino-3,6,9,12-tetraoxatetradecyl)-2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetamide hydrochloride;Thalidomide-O-amido-PEG4-NH2 hydrochloride;Thalidomide-O-C1-amido-PEG4-C2-NH2 HCl;Acetamide,?N-(14-amino-3,6,9,12-tetraoxatetradec-1-yl)-2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]oxy]-, hydrochloride (1:1);Thalidomide-O-amido-PEG4-C2-NH2 HC;Thalidomide-O-amido-PEG4-C2-NH2 HCl
CAS:2245697-85-0
MF:C25H35ClN4O10
MW:587.02
EINECS:
Product Categories:
Mol File:2245697-85-0.mol
Thalidomide-O-amido-PEG4-C2-NH2 hydrochloride Structure
Thalidomide-O-amido-PEG4-C2-NH2 hydrochloride Chemical Properties
storage temp. 2-8°C, sealed storage, away from moisture
solubility Soluble in DMSO
form Oil
color Light yellow to yellow
Safety Information
MSDS Information
Thalidomide-O-amido-PEG4-C2-NH2 hydrochloride Usage And Synthesis
UsesThalidomide-O-amido-PEG4-C2-NH2 hydrochloride, a synthesized E3 ligase ligand-linker conjugate that incorporates the Thalidomide based cereblon ligand and a linker, can be used in the synthesis of PROTACs[1].
IC 50Cereblon
storageStore at -20°C
References[1] James Bradner, et al. Methods to induce targeted protein degradation through bifunctional molecules. WO2016105518A1.
Thalidomide-O-amido-PEG4-C2-NH2 hydrochloride Preparation Products And Raw materials
Tag:Thalidomide-O-amido-PEG4-C2-NH2 hydrochloride(2245697-85-0) Related Product Information
Thalidomide-O-amido-PEG4-azide Thalidomide-linker 14 Thalidomide-linker 13 N-(4-azidobutyl)-2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetamide E3 Ligase Ligand-Linker Conjugates 20 Thalidomide-O-C6-NH2 TFA Thalidomide-O-amido-C4-NH2 hydrochloride Thalidomide-O-amido-PEG3-C2-NH2 hydrochloride Thalidomide-O-amido-C3-NH2 (TFA) E3 Ligase Ligand-Linker Conjugates 21 E3 Ligase Ligand-Linker Conjugates 19 Thalidomide-linker 15 Thalidomide-O-amido-C8-NH2 hydrochloride Thalidomide-O-amido-PEG1-(C1-?PEG)2-C2-NH2 N-(3-(2-(2-(3-Aminopropoxy)ethoxy)ethoxy)propyl)-2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetamide Trifluoroacetate E3 Ligase Ligand-Linker Conjugates 24 (TFA) Thalidomide-O-C6-NH2 Acetamide, N-(5-aminopentyl)-2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]oxy]-